Wilkinson SM - Search Results

1

Pharmacological Evaluation of Novel Bioisosteres of an Adamantanyl Benzamide P2X₇ Receptor Antagonist.

Wilkinson SM, Barron ML, O'Brien-Brown J, Janssen B, Stokes L, Werry EL, Chishty M, Skarratt KK, Ong JA, Hibbs DE, Vugts DJ, Fuller S, Windhorst AD, Kassiou M. Wilkinson SM, et al. ACS Chem Neurosci. 2017 Nov 15;8(11):2374-2380. doi: 10.1021/acschemneuro.7b00272. Epub 2017 Aug 25. ACS Chem Neurosci. 2017. PMID: 28841278

2

Identification of the allosteric P2X₇ receptor antagonist [¹¹C]SMW139 as a PET tracer of microglial activation.

Janssen B, Vugts DJ, Wilkinson SM, Ory D, Chalon S, Hoozemans JJM, Schuit RC, Beaino W, Kooijman EJM, van den Hoek J, Chishty M, Doméné A, Van der Perren A, Villa A, Maggi A, Molenaar GT, Funke U, Shevchenko RV, Baekelandt V, Bormans G, Lammertsma AA, Kassiou M, Windhorst AD. Janssen B, et al. Among authors: wilkinson sm. Sci Rep. 2018 Apr 26;8(1):6580. doi: 10.1038/s41598-018-24814-0. Sci Rep. 2018. PMID: 29700413 Free PMC article.

3

Discovery and pharmacological evaluation of a novel series of adamantyl cyanoguanidines as P2X₇ receptor antagonists.

O'Brien-Brown J, Jackson A, Reekie TA, Barron ML, Werry EL, Schiavini P, McDonnell M, Munoz L, Wilkinson S, Noll B, Wang S, Kassiou M. O'Brien-Brown J, et al. Eur J Med Chem. 2017 Apr 21;130:433-439. doi: 10.1016/j.ejmech.2017.02.060. Epub 2017 Mar 2. Eur J Med Chem. 2017. PMID: 28279849

4

Effects of bioisosteric fluorine in synthetic cannabinoid designer drugs JWH-018, AM-2201, UR-144, XLR-11, PB-22, 5F-PB-22, APICA, and STS-135.

Banister SD, Stuart J, Kevin RC, Edington A, Longworth M, Wilkinson SM, Beinat C, Buchanan AS, Hibbs DE, Glass M, Connor M, McGregor IS, Kassiou M. Banister SD, et al. Among authors: wilkinson sm. ACS Chem Neurosci. 2015 Aug 19;6(8):1445-58. doi: 10.1021/acschemneuro.5b00107. Epub 2015 May 8. ACS Chem Neurosci. 2015. PMID: 25921407

5

The synthesis and pharmacological evaluation of adamantane-derived indoles: cannabimimetic drugs of abuse.

Banister SD, Wilkinson SM, Longworth M, Stuart J, Apetz N, English K, Brooker L, Goebel C, Hibbs DE, Glass M, Connor M, McGregor IS, Kassiou M. Banister SD, et al. Among authors: wilkinson sm. ACS Chem Neurosci. 2013 Jul 17;4(7):1081-92. doi: 10.1021/cn400035r. Epub 2013 Apr 17. ACS Chem Neurosci. 2013. PMID: 23551277 Free PMC article.

6

The first CNS-active carborane: A novel P2X7 receptor antagonist with antidepressant activity.

Wilkinson SM, Gunosewoyo H, Barron ML, Boucher A, McDonnell M, Turner P, Morrison DE, Bennett MR, McGregor IS, Rendina LM, Kassiou M. Wilkinson SM, et al. ACS Chem Neurosci. 2014 May 21;5(5):335-9. doi: 10.1021/cn500054n. Epub 2014 Apr 3. ACS Chem Neurosci. 2014. PMID: 24689484 Free PMC article. Review.

7

Pharmacological characterization of a structural hybrid P2X7R antagonist using ATP and LL-37.

Jackson A, Werry EL, O'Brien-Brown J, Schiavini P, Wilkinson S, Wong ECN, McKenzie ADJ, Maximova A, Kassiou M. Jackson A, et al. Eur J Pharmacol. 2022 Jan 5;914:174667. doi: 10.1016/j.ejphar.2021.174667. Epub 2021 Dec 1. Eur J Pharmacol. 2022. PMID: 34863711

8

Pharmacology of Indole and Indazole Synthetic Cannabinoid Designer Drugs AB-FUBINACA, ADB-FUBINACA, AB-PINACA, ADB-PINACA, 5F-AB-PINACA, 5F-ADB-PINACA, ADBICA, and 5F-ADBICA.

Banister SD, Moir M, Stuart J, Kevin RC, Wood KE, Longworth M, Wilkinson SM, Beinat C, Buchanan AS, Glass M, Connor M, McGregor IS, Kassiou M. Banister SD, et al. Among authors: wilkinson sm. ACS Chem Neurosci. 2015 Sep 16;6(9):1546-59. doi: 10.1021/acschemneuro.5b00112. Epub 2015 Jul 17. ACS Chem Neurosci. 2015. PMID: 26134475

9

Rapid access to N-(indol-2-yl)amides and N-(indol-3-yl)amides as unexplored pharmacophores.

Reekie TA, Wilkinson SM, Law V, Hibbs DE, Ong JA, Kassiou M. Reekie TA, et al. Among authors: wilkinson sm. Org Biomol Chem. 2017 Jan 18;15(3):576-580. doi: 10.1039/c6ob02622b. Org Biomol Chem. 2017. PMID: 27991628

10

A systematic exploration of the effects of flexibility and basicity on sigma (σ) receptor binding in a series of substituted diamines.

Conroy T, Manohar M, Gong Y, Wilkinson SM, Webster M, Lieberman BP, Banister SD, Reekie TA, Mach RH, Rendina LM, Kassiou M. Conroy T, et al. Among authors: wilkinson sm. Org Biomol Chem. 2016 Oct 4;14(39):9388-9405. doi: 10.1039/c6ob00615a. Org Biomol Chem. 2016. PMID: 27714195

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