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CYP-Mediated Sulfoximine Deimination of AZD6738.
Drug Metab Dispos. 2017 Nov;45(11):1133-1138. doi: 10.1124/dmd.117.077776. Epub 2017 Aug 23.
Drug Metab Dispos. 2017.
PMID: 28835442
Impact of Interindividual Differences in Plasma Fraction Unbound on the Pharmacokinetics of a Novel Syk Kinase Inhibitor in Beagle Dogs.
Pike A, Jones B, Markandu R, O'Neill D.
Pike A, et al. Among authors: markandu r.
Drug Metab Dispos. 2021 Sep;49(9):736-742. doi: 10.1124/dmd.121.000409. Epub 2021 Jun 16.
Drug Metab Dispos. 2021.
PMID: 34135088
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Drug metabolite identification using ultrahigh-performance liquid chromatography-ultraviolet spectroscopy and parallelized scans on a tribrid Orbitrap mass spectrometer.
Wilkinson SD, Martin S, Orton AL, Markandu R, Jones BC.
Wilkinson SD, et al. Among authors: markandu r.
Rapid Commun Mass Spectrom. 2020 May 30;34(10):e8735. doi: 10.1002/rcm.8735.
Rapid Commun Mass Spectrom. 2020.
PMID: 31967694
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Optimization of an Imidazo[1,2-a]pyridine Series to Afford Highly Selective Type I1/2 Dual Mer/Axl Kinase Inhibitors with In Vivo Efficacy.
McCoull W, Boyd S, Brown MR, Coen M, Collingwood O, Davies NL, Doherty A, Fairley G, Goldberg K, Hardaker E, He G, Hennessy EJ, Hopcroft P, Hodgson G, Jackson A, Jiang X, Karmokar A, Lainé AL, Lindsay N, Mao Y, Markandu R, McMurray L, McLean N, Mooney L, Musgrove H, Nissink JWM, Pflug A, Reddy VP, Rawlins PB, Rivers E, Schimpl M, Smith GF, Tentarelli S, Travers J, Troup RI, Walton J, Wang C, Wilkinson S, Williamson B, Winter-Holt J, Yang D, Zheng Y, Zhu Q, Smith PD.
McCoull W, et al. Among authors: markandu r.
J Med Chem. 2021 Sep 23;64(18):13524-13539. doi: 10.1021/acs.jmedchem.1c00920. Epub 2021 Sep 3.
J Med Chem. 2021.
PMID: 34478292
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Development of a quantification method for arginase inhibitors by LC-MS/MS with benzoyl chloride derivatization.
Gosselin E, Pop-Damkov P, Xue A, Markandu R, Mlynarski S, Finlay R, Schuller A, Ramsden D, Gangl ET.
Gosselin E, et al. Among authors: markandu r.
J Pharm Biomed Anal. 2024 May 8;246:116210. doi: 10.1016/j.jpba.2024.116210. Online ahead of print.
J Pharm Biomed Anal. 2024.
PMID: 38788624
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