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Thiosemicarbazones and 4-thiazolidinones indole-based derivatives: Synthesis, evaluation of antiproliferative activity, cell death mechanisms and topoisomerase inhibition assay.
de Oliveira JF, Lima TS, Vendramini-Costa DB, de Lacerda Pedrosa SCB, Lafayette EA, da Silva RMF, de Almeida SMV, de Moura RO, Ruiz ALTG, de Carvalho JE, de Lima MDCA. de Oliveira JF, et al. Among authors: de almeida smv, de moura ro, de lacerda pedrosa scb, de carvalho je, de lima mdca. Eur J Med Chem. 2017 Aug 18;136:305-314. doi: 10.1016/j.ejmech.2017.05.023. Epub 2017 May 8. Eur J Med Chem. 2017. PMID: 28505535
Synthesis, cytotoxicity and antifungal activity of 5-nitro-thiophene-thiosemicarbazones derivatives.
de Araújo Neto LN, do Carmo Alves de Lima M, de Oliveira JF, de Souza ER, Buonafina MDS, Vitor Anjos MN, Brayner FA, Alves LC, Neves RP, Mendonça-Junior FJB. de Araújo Neto LN, et al. Among authors: de souza er, de oliveira jf. Chem Biol Interact. 2017 Jun 25;272:172-181. doi: 10.1016/j.cbi.2017.05.005. Epub 2017 May 4. Chem Biol Interact. 2017. PMID: 28479098 Free article.
Medicinal chemistry of antischistosomal drugs: Praziquantel and oxamniquine.
da Silva VBR, Campos BRKL, de Oliveira JF, Decout JL, do Carmo Alves de Lima M. da Silva VBR, et al. Among authors: de oliveira jf. Bioorg Med Chem. 2017 Jul 1;25(13):3259-3277. doi: 10.1016/j.bmc.2017.04.031. Epub 2017 Apr 27. Bioorg Med Chem. 2017. PMID: 28495384 Review.
Synthesis and in vitro anticancer activity of new 2-thioxo-oxazolidin-4-one derivatives.
Campos JF, Pereira MC, de Sena WLB, de Barros Martins CG, de Oliveira JF, da Cruz Amorim CA, de Melo Rêgo MJB, da Rocha Pitta MG, de Lima MDCA, da Rocha Pitta MG, da Rocha Pitta I. Campos JF, et al. Among authors: de sena wlb, de melo rego mjb, de barros martins cg, de oliveira jf, de lima mdca. Pharmacol Rep. 2017 Aug;69(4):633-641. doi: 10.1016/j.pharep.2017.03.005. Epub 2017 Mar 18. Pharmacol Rep. 2017. PMID: 28511054
Synthesis of novel indole derivatives as promising DNA-binding agents and evaluation of antitumor and antitopoisomerase I activities.
Lafayette EA, de Almeida SMV, Cavalcanti Santos RV, de Oliveira JF, Amorim CADC, da Silva RMF, Pitta MGDR, Pitta IDR, de Moura RO, de Carvalho Júnior LB, de Melo Rêgo MJB, de Lima MDCA. Lafayette EA, et al. Among authors: de almeida smv, de moura ro, de carvalho junior lb, de melo rego mjb, de oliveira jf, de lima mdca. Eur J Med Chem. 2017 Aug 18;136:511-522. doi: 10.1016/j.ejmech.2017.05.012. Epub 2017 May 4. Eur J Med Chem. 2017. PMID: 28531811
DNA binding and Topoisomerase inhibition: How can these mechanisms be explored to design more specific anticancer agents?
de Almeida SMV, Ribeiro AG, de Lima Silva GC, Ferreira Alves JE, Beltrão EIC, de Oliveira JF, de Carvalho LB Junior, Alves de Lima MDC. de Almeida SMV, et al. Among authors: de carvalho lb junior, de lima silva gc, de oliveira jf. Biomed Pharmacother. 2017 Dec;96:1538-1556. doi: 10.1016/j.biopha.2017.11.054. Epub 2017 Nov 22. Biomed Pharmacother. 2017. PMID: 29174576 Review.
New 1,3-benzodioxole derivatives: Synthesis, evaluation of in vitro schistosomicidal activity and ultrastructural analysis.
Mariz Gomes da Silva LM, de Oliveira JF, Silva WL, da Silva AL, de Almeida Junior ASA, Barbosa Dos Santos VH, Alves LC, Brayner Dos Santos FA, Costa VMA, Aires AL, de Lima MDCA, Albuquerque MCPA. Mariz Gomes da Silva LM, et al. Among authors: de almeida junior asa, de oliveira jf, de lima mdca. Chem Biol Interact. 2018 Mar 1;283:20-29. doi: 10.1016/j.cbi.2018.01.016. Epub 2018 Jan 31. Chem Biol Interact. 2018. PMID: 29366735 Free article.
New thiophene-acridine compounds: Synthesis, antileishmanial activity, DNA binding, chemometric, and molecular docking studies.
de Lima Serafim V, Félix MB, Frade Silva DK, Rodrigues KADF, Andrade PN, de Almeida SMV, de Albuquerque Dos Santos S, de Oliveira JF, de Lima MDCA, Mendonça-Junior FJB, Scotti MT, de Oliveira MR, de Moura RO. de Lima Serafim V, et al. Among authors: de almeida smv, de moura ro, de albuquerque dos santos s, de oliveira mr, de oliveira jf, de lima mdca. Chem Biol Drug Des. 2018 Jun;91(6):1141-1155. doi: 10.1111/cbdd.13176. Epub 2018 Mar 25. Chem Biol Drug Des. 2018. PMID: 29415325
139 results