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Modulating 5-HT4 and 5-HT6 receptors in Alzheimer's disease treatment.
Future Med Chem. 2017 May;9(8):781-795. doi: 10.4155/fmc-2017-0031. Epub 2017 May 15.
Future Med Chem. 2017.
PMID: 28504917
Review.
Synthesis and evaluation of novel serotonin 4 receptor radiotracers for single photon emission computed tomography.
Lalut J, Tournier BB, Cailly T, Lecoutey C, Corvaisier S, Davis A, Ballandonne C, Since M, Millet P, Fabis F, Dallemagne P, Rochais C.
Lalut J, et al.
Eur J Med Chem. 2016 Jun 30;116:90-101. doi: 10.1016/j.ejmech.2016.03.059. Epub 2016 Mar 25.
Eur J Med Chem. 2016.
PMID: 27060761
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Novel multitarget-directed ligands targeting acetylcholinesterase and σ1 receptors as lead compounds for treatment of Alzheimer's disease: Synthesis, evaluation, and structural characterization of their complexes with acetylcholinesterase.
Lalut J, Santoni G, Karila D, Lecoutey C, Davis A, Nachon F, Silman I, Sussman J, Weik M, Maurice T, Dallemagne P, Rochais C.
Lalut J, et al.
Eur J Med Chem. 2019 Jan 15;162:234-248. doi: 10.1016/j.ejmech.2018.10.064. Epub 2018 Nov 8.
Eur J Med Chem. 2019.
PMID: 30447434
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Inhibiting Acetylcholinesterase to Activate Pleiotropic Prodrugs with Therapeutic Interest in Alzheimer's Disease.
Toublet FX, Lecoutey C, Lalut J, Hatat B, Davis A, Since M, Corvaisier S, Freret T, Sopkova de Oliveira Santos J, Claeysen S, Boulouard M, Dallemagne P, Rochais C.
Toublet FX, et al. Among authors: lalut j.
Molecules. 2019 Jul 31;24(15):2786. doi: 10.3390/molecules24152786.
Molecules. 2019.
PMID: 31370232
Free PMC article.
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Rational design of novel benzisoxazole derivatives with acetylcholinesterase inhibitory and serotoninergic 5-HT4 receptors activities for the treatment of Alzheimer's disease.
Lalut J, Payan H, Davis A, Lecoutey C, Legay R, Sopkova-de Oliveira Santos J, Claeysen S, Dallemagne P, Rochais C.
Lalut J, et al.
Sci Rep. 2020 Feb 20;10(1):3014. doi: 10.1038/s41598-020-59805-7.
Sci Rep. 2020.
PMID: 32080261
Free PMC article.
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Pleiotropic prodrugs: Design of a dual butyrylcholinesterase inhibitor and 5-HT6 receptor antagonist with therapeutic interest in Alzheimer's disease.
Toublet FX, Lalut J, Hatat B, Lecoutey C, Davis A, Since M, Corvaisier S, Freret T, Sopková-de Oliveira Santos J, Claeysen S, Boulouard M, Dallemagne P, Rochais C.
Toublet FX, et al. Among authors: lalut j.
Eur J Med Chem. 2021 Jan 15;210:113059. doi: 10.1016/j.ejmech.2020.113059. Epub 2020 Dec 3.
Eur J Med Chem. 2021.
PMID: 33310288
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Synthesis of C3-arylated-3-deazauridine derivatives with potent anti-HSV-1 activities.
Lalut J, Tripoteau L, Marty C, Bares H, Bourgougnon N, Felpin FX.
Lalut J, et al.
Bioorg Med Chem Lett. 2012 Dec 15;22(24):7461-4. doi: 10.1016/j.bmcl.2012.10.047. Epub 2012 Oct 24.
Bioorg Med Chem Lett. 2012.
PMID: 23141915
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