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Medicinal chemistry of antischistosomal drugs: Praziquantel and oxamniquine.
da Silva VBR, Campos BRKL, de Oliveira JF, Decout JL, do Carmo Alves de Lima M. da Silva VBR, et al. Among authors: de oliveira jf. Bioorg Med Chem. 2017 Jul 1;25(13):3259-3277. doi: 10.1016/j.bmc.2017.04.031. Epub 2017 Apr 27. Bioorg Med Chem. 2017. PMID: 28495384 Review.
Synthesis, cytotoxicity and antifungal activity of 5-nitro-thiophene-thiosemicarbazones derivatives.
de Araújo Neto LN, do Carmo Alves de Lima M, de Oliveira JF, de Souza ER, Buonafina MDS, Vitor Anjos MN, Brayner FA, Alves LC, Neves RP, Mendonça-Junior FJB. de Araújo Neto LN, et al. Among authors: de souza er, de oliveira jf. Chem Biol Interact. 2017 Jun 25;272:172-181. doi: 10.1016/j.cbi.2017.05.005. Epub 2017 May 4. Chem Biol Interact. 2017. PMID: 28479098 Free article.
Thiosemicarbazones and 4-thiazolidinones indole-based derivatives: Synthesis, evaluation of antiproliferative activity, cell death mechanisms and topoisomerase inhibition assay.
de Oliveira JF, Lima TS, Vendramini-Costa DB, de Lacerda Pedrosa SCB, Lafayette EA, da Silva RMF, de Almeida SMV, de Moura RO, Ruiz ALTG, de Carvalho JE, de Lima MDCA. de Oliveira JF, et al. Among authors: de almeida smv, de moura ro, de lacerda pedrosa scb, de carvalho je, de lima mdca. Eur J Med Chem. 2017 Aug 18;136:305-314. doi: 10.1016/j.ejmech.2017.05.023. Epub 2017 May 8. Eur J Med Chem. 2017. PMID: 28505535
Synthesis of novel indole derivatives as promising DNA-binding agents and evaluation of antitumor and antitopoisomerase I activities.
Lafayette EA, de Almeida SMV, Cavalcanti Santos RV, de Oliveira JF, Amorim CADC, da Silva RMF, Pitta MGDR, Pitta IDR, de Moura RO, de Carvalho Júnior LB, de Melo Rêgo MJB, de Lima MDCA. Lafayette EA, et al. Among authors: de almeida smv, de moura ro, de carvalho junior lb, de melo rego mjb, de oliveira jf, de lima mdca. Eur J Med Chem. 2017 Aug 18;136:511-522. doi: 10.1016/j.ejmech.2017.05.012. Epub 2017 May 4. Eur J Med Chem. 2017. PMID: 28531811
Synthesis, DNA and protein interactions and human topoisomerase inhibition of novel Spiroacridine derivatives.
Gouveia RG, Ribeiro AG, Segundo MÂSP, de Oliveira JF, de Lima MDCA, de Lima Souza TRC, de Almeida SMV, de Moura RO. Gouveia RG, et al. Among authors: de almeida smv, de moura ro, de lima souza trc, de oliveira jf, de lima mdca. Bioorg Med Chem. 2018 Dec 1;26(22):5911-5921. doi: 10.1016/j.bmc.2018.10.038. Epub 2018 Oct 29. Bioorg Med Chem. 2018. PMID: 30420325
In vitro activity, ultrastructural studies and in silico pharmacokinetic properties of indol-3-yl-thiosemicarbazones derivatives and analogues against juvenile and adult worms of S. mansoni.
de Almeida Júnior ASA, de Oliveira JF, da Silva AL, da Rocha RET, Junior NCP, Gouveia ALA, da Silva RMF, de Azevedo Albuquerque MCP, Brayner FA, Alves LC, do Carmo Alves de Lima M. de Almeida Júnior ASA, et al. Among authors: de azevedo albuquerque mcp, de oliveira jf. Eur J Pharm Sci. 2019 Oct 1;138:104985. doi: 10.1016/j.ejps.2019.104985. Epub 2019 Jul 5. Eur J Pharm Sci. 2019. PMID: 31283945
Thiazolidinedione and thiazole derivatives potentiate norfloxacin activity against NorA efflux pump over expression in Staphylococcus aureus 1199B strains.
Pereira PS, Lima MDCA, Neto PPM, Oliveira-Tintino CDM, Tintino SR, Menezes IRA, de Oliveira JF, Marchand P, Coutinho HDM, Rodrigues MDD, da Silva TG. Pereira PS, et al. Among authors: oliveira tintino cdm, de oliveira jf. Bioorg Med Chem. 2019 Sep 1;27(17):3797-3804. doi: 10.1016/j.bmc.2019.07.006. Epub 2019 Jul 4. Bioorg Med Chem. 2019. PMID: 31320212 Free article.
Topoisomerase inhibition and albumin interaction studies of acridine-thiosemicarbazone derivatives.
da Silva Filho FA, de Freitas Souza T, Ribeiro AG, Alves JEF, de Oliveira JF, de Lima Souza TRC, de Moura RO, do Carmo Alves de Lima M, de Carvalho Junior LB, de Almeida SMV. da Silva Filho FA, et al. Among authors: de almeida smv, de moura ro, de carvalho junior lb, de freitas souza t, de lima souza trc, de oliveira jf. Int J Biol Macromol. 2019 Oct 1;138:582-589. doi: 10.1016/j.ijbiomac.2019.07.097. Epub 2019 Jul 16. Int J Biol Macromol. 2019. PMID: 31323270 Free article.
Novel 4-quinoline-thiosemicarbazone derivatives: Synthesis, antiproliferative activity, in vitro and in silico biomacromolecule interaction studies and topoisomerase inhibition.
Ribeiro AG, Almeida SMV, de Oliveira JF, Souza TRCL, Santos KLD, Albuquerque APB, Nogueira MCBL, Carvalho Junior LB, Moura RO, da Silva AC, Pereira VRA, Castro MCAB, Lima MDCA. Ribeiro AG, et al. Among authors: de oliveira jf. Eur J Med Chem. 2019 Nov 15;182:111592. doi: 10.1016/j.ejmech.2019.111592. Epub 2019 Aug 6. Eur J Med Chem. 2019. PMID: 31421632
139 results