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Functional, thermodynamics, structural and biological studies of in silico-identified inhibitors of Mycobacterium tuberculosis enoyl-ACP(CoA) reductase enzyme.
Sci Rep. 2017 Apr 24;7:46696. doi: 10.1038/srep46696.
Sci Rep. 2017.
PMID: 28436453
Free PMC article.
Mefloquine and its oxazolidine derivative compound are active against drug-resistant Mycobacterium tuberculosis strains and in a murine model of tuberculosis infection.
Rodrigues-Junior VS, Villela AD, Gonçalves RS, Abbadi BL, Trindade RV, López-Gavín A, Tudó G, González-Martín J, Basso LA, de Souza MV, Campos MM, Santos DS.
Rodrigues-Junior VS, et al. Among authors: trindade rv.
Int J Antimicrob Agents. 2016 Aug;48(2):203-7. doi: 10.1016/j.ijantimicag.2016.04.029. Epub 2016 Jun 7.
Int J Antimicrob Agents. 2016.
PMID: 27364701
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New insights into the SAR and drug combination synergy of 2-(quinolin-4-yloxy)acetamides against Mycobacterium tuberculosis.
Giacobbo BC, Pissinate K, Rodrigues-Junior V, Villela AD, Grams ES, Abbadi BL, Subtil FT, Sperotto N, Trindade RV, Back DF, Campos MM, Basso LA, Machado P, Santos DS.
Giacobbo BC, et al. Among authors: trindade rv.
Eur J Med Chem. 2017 Jan 27;126:491-501. doi: 10.1016/j.ejmech.2016.11.048. Epub 2016 Nov 23.
Eur J Med Chem. 2017.
PMID: 27914363
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Pulse Proteolysis and Precipitation for Target Identification.
Trindade RV, Pinto AF, Santos DS, Bizarro CV.
Trindade RV, et al.
J Proteome Res. 2016 Jul 1;15(7):2236-45. doi: 10.1021/acs.jproteome.6b00214. Epub 2016 Jun 20.
J Proteome Res. 2016.
PMID: 27255303
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2-(Quinolin-4-yloxy)acetamides Are Active against Drug-Susceptible and Drug-Resistant Mycobacterium tuberculosis Strains.
Pissinate K, Villela AD, Rodrigues-Junior V, Giacobbo BC, Grams ES, Abbadi BL, Trindade RV, Roesler Nery L, Bonan CD, Back DF, Campos MM, Basso LA, Santos DS, Machado P.
Pissinate K, et al. Among authors: trindade rv.
ACS Med Chem Lett. 2016 Jan 11;7(3):235-9. doi: 10.1021/acsmedchemlett.5b00324. eCollection 2016 Mar 10.
ACS Med Chem Lett. 2016.
PMID: 26985307
Free PMC article.
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