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RGD-mediated delivery of small-molecule drugs.
Future Med Chem. 2017 Apr;9(6):579-604. doi: 10.4155/fmc-2017-0008. Epub 2017 Apr 10.
Future Med Chem. 2017.
PMID: 28394627
Review.
Synthesis and biological evaluation of a Platinum(II)-c(RGDyK) conjugate for integrin-targeted photodynamic therapy.
Chatzisideri T, Thysiadis S, Katsamakas S, Dalezis P, Sigala I, Lazarides T, Nikolakaki E, Trafalis D, Gederaas OA, Lindgren M, Sarli V.
Chatzisideri T, et al.
Eur J Med Chem. 2017 Dec 1;141:221-231. doi: 10.1016/j.ejmech.2017.09.058. Epub 2017 Sep 28.
Eur J Med Chem. 2017.
PMID: 29031069
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Novel c(RGDyK)-based conjugates of POPAM and 5-fluorouracil for integrin-targeted cancer therapy.
Thysiadis S, Katsamakas S, Dalezis P, Chatzisideri T, Trafalis D, Sarli V.
Thysiadis S, et al. Among authors: chatzisideri t.
Future Med Chem. 2017 Dec;9(18):2181-2196. doi: 10.4155/fmc-2017-0139. Epub 2017 Nov 7.
Future Med Chem. 2017.
PMID: 29110537
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Cancer-targeted delivery systems based on peptides.
Chatzisideri T, Leonidis G, Sarli V.
Chatzisideri T, et al.
Future Med Chem. 2018 Sep 1;10(18):2201-2226. doi: 10.4155/fmc-2018-0174. Epub 2018 Jul 25.
Future Med Chem. 2018.
PMID: 30043641
Review.
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Synthesis and biological studies of c(RGDyK) conjugates of cucurbitacins.
Chatzisideri T, Dalezis P, Leonidis G, Bousis S, Trafalis D, Bianchini F, Sarli V.
Chatzisideri T, et al.
Future Med Chem. 2021 May;13(10):877-895. doi: 10.4155/fmc-2020-0309. Epub 2021 Apr 16.
Future Med Chem. 2021.
PMID: 33858195
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Integrin-Mediated Targeted Cancer Therapy Using c(RGDyK)-Based Conjugates of Gemcitabine.
Chatzisideri T, Leonidis G, Karampelas T, Skavatsou E, Velentza-Almpani A, Bianchini F, Tamvakopoulos C, Sarli V.
Chatzisideri T, et al.
J Med Chem. 2022 Jan 13;65(1):271-284. doi: 10.1021/acs.jmedchem.1c01468. Epub 2021 Dec 30.
J Med Chem. 2022.
PMID: 34967607
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