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Structure-Activity Relationship of the Antimalarial Ozonide Artefenomel (OZ439).
J Med Chem. 2017 Apr 13;60(7):2654-2668. doi: 10.1021/acs.jmedchem.6b01586. Epub 2017 Jan 18.
J Med Chem. 2017.
PMID: 28052200
Structure-Activity Relationship of Antischistosomal Ozonide Carboxylic Acids.
Wu J, Wang X, Chiu FCK, Häberli C, Shackleford DM, Ryan E, Kamaraj S, Bulbule VJ, Wallick AI, Dong Y, White KL, Davis PH, Charman SA, Keiser J, Vennerstrom JL.
Wu J, et al. Among authors: bulbule vj.
J Med Chem. 2020 Apr 9;63(7):3723-3736. doi: 10.1021/acs.jmedchem.0c00069. Epub 2020 Mar 19.
J Med Chem. 2020.
PMID: 32134263
Free PMC article.
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Second generation tetrahydroquinoline-based protein farnesyltransferase inhibitors as antimalarials.
Bendale P, Olepu S, Suryadevara PK, Bulbule V, Rivas K, Nallan L, Smart B, Yokoyama K, Ankala S, Pendyala PR, Floyd D, Lombardo LJ, Williams DK, Buckner FS, Chakrabarti D, Verlinde CL, Van Voorhis WC, Gelb MH.
Bendale P, et al.
J Med Chem. 2007 Sep 20;50(19):4585-605. doi: 10.1021/jm0703340. Epub 2007 Aug 28.
J Med Chem. 2007.
PMID: 17722901
Free PMC article.
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2-Oxotetrahydroquinoline-based antimalarials with high potency and metabolic stability.
Bulbule VJ, Rivas K, Verlinde CL, Van Voorhis WC, Gelb MH.
Bulbule VJ, et al.
J Med Chem. 2008 Feb 14;51(3):384-7. doi: 10.1021/jm7013138. Epub 2008 Jan 17.
J Med Chem. 2008.
PMID: 18198825
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