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Page 1
Efflux Pump Blockers in Gram-Negative Bacteria: The New Generation of Hydantoin Based-Modulators to Improve Antibiotic Activity.
Otręebska-Machaj E, Chevalier J, Handzlik J, Szymańska E, Schabikowski J, Boyer G, Bolla JM, Kieć-Kononowicz K, Pagès JM, Alibert S. Otręebska-Machaj E, et al. Among authors: schabikowski j. Front Microbiol. 2016 May 3;7:622. doi: 10.3389/fmicb.2016.00622. eCollection 2016. Front Microbiol. 2016. PMID: 27199950 Free PMC article.
Imidazolidine-4-one derivatives in the search for novel chemosensitizers of Staphylococcus aureus MRSA: synthesis, biological evaluation and molecular modeling studies.
Matys A, Podlewska S, Witek K, Witek J, Bojarski AJ, Schabikowski J, Otrębska-Machaj E, Latacz G, Szymańska E, Kieć-Kononowicz K, Molnar J, Amaral L, Handzlik J. Matys A, et al. Among authors: schabikowski j. Eur J Med Chem. 2015 Aug 28;101:313-25. doi: 10.1016/j.ejmech.2015.06.013. Epub 2015 Jun 24. Eur J Med Chem. 2015. PMID: 26160112
Similarities and differences in affinity and binding modes of tricyclic pyrimido- and pyrazinoxanthines at human and rat adenosine receptors.
Szymańska E, Drabczyńska A, Karcz T, Müller CE, Köse M, Karolak-Wojciechowska J, Fruziński A, Schabikowski J, Doroz-Płonka A, Handzlik J, Kieć-Kononowicz K. Szymańska E, et al. Among authors: schabikowski j. Bioorg Med Chem. 2016 Sep 15;24(18):4347-4362. doi: 10.1016/j.bmc.2016.07.028. Epub 2016 Jul 18. Bioorg Med Chem. 2016. PMID: 27485602
Tricyclic xanthine derivatives containing a basic substituent: adenosine receptor affinity and drug-related properties.
Załuski M, Stanuch K, Karcz T, Hinz S, Latacz G, Szymańska E, Schabikowski J, Doroż-Płonka A, Handzlik J, Drabczyńska A, Müller CE, Kieć-Kononowicz K. Załuski M, et al. Among authors: schabikowski j. Medchemcomm. 2018 May 14;9(6):951-962. doi: 10.1039/c8md00070k. eCollection 2018 Jun 1. Medchemcomm. 2018. PMID: 30108984 Free PMC article.
Novel multi-target directed ligands based on annelated xanthine scaffold with aromatic substituents acting on adenosine receptor and monoamine oxidase B. Synthesis, in vitro and in silico studies.
Załuski M, Schabikowski J, Schlenk M, Olejarz-Maciej A, Kubas B, Karcz T, Kuder K, Latacz G, Zygmunt M, Synak D, Hinz S, Müller CE, Kieć-Kononowicz K. Załuski M, et al. Among authors: schabikowski j. Bioorg Med Chem. 2019 Apr 1;27(7):1195-1210. doi: 10.1016/j.bmc.2019.02.004. Epub 2019 Feb 2. Bioorg Med Chem. 2019. PMID: 30808606
Antiplatelet Effects of Selected Xanthine-Based Adenosine A2A and A2B Receptor Antagonists Determined in Rat Blood.
Kubacka M, Mogilski S, Bednarski M, Pociecha K, Świerczek A, Nicosia N, Schabikowski J, Załuski M, Chłoń-Rzepa G, Hockemeyer J, Müller CE, Kieć-Kononowicz K, Kotańska M. Kubacka M, et al. Among authors: schabikowski j. Int J Mol Sci. 2023 Aug 29;24(17):13378. doi: 10.3390/ijms241713378. Int J Mol Sci. 2023. PMID: 37686188 Free PMC article.
8-Benzylaminoxanthine scaffold variations for selective ligands acting on adenosine A2A receptors. Design, synthesis and biological evaluation.
Załuski M, Schabikowski J, Jaśko P, Bryła A, Olejarz-Maciej A, Kaleta M, Głuch-Lutwin M, Brockmann A, Hinz S, Zygmunt M, Kuder K, Latacz G, Vielmuth C, Müller CE, Kieć-Kononowicz K. Załuski M, et al. Among authors: schabikowski j. Bioorg Chem. 2020 Aug;101:104033. doi: 10.1016/j.bioorg.2020.104033. Epub 2020 Jun 19. Bioorg Chem. 2020. PMID: 32629282
A2B Adenosine Receptor Antagonists with Picomolar Potency.
Jiang J, Seel CJ, Temirak A, Namasivayam V, Arridu A, Schabikowski J, Baqi Y, Hinz S, Hockemeyer J, Müller CE. Jiang J, et al. Among authors: schabikowski j. J Med Chem. 2019 Apr 25;62(8):4032-4055. doi: 10.1021/acs.jmedchem.9b00071. Epub 2019 Apr 15. J Med Chem. 2019. PMID: 30835463