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Molecular Basis of Valine-Citrulline-PABC Linker Instability in Site-Specific ADCs and Its Mitigation by Linker Design.
Mol Cancer Ther. 2016 May;15(5):958-70. doi: 10.1158/1535-7163.MCT-15-1004. Epub 2016 Mar 4.
Mol Cancer Ther. 2016.
PMID: 26944918
Site-specific conjugation improves therapeutic index of antibody drug conjugates with high drug loading.
Strop P, Delaria K, Foletti D, Witt JM, Hasa-Moreno A, Poulsen K, Casas MG, Dorywalska M, Farias S, Pios A, Lui V, Dushin R, Zhou D, Navaratnam T, Tran TT, Sutton J, Lindquist KC, Han B, Liu SH, Shelton DL, Pons J, Rajpal A.
Strop P, et al. Among authors: navaratnam t.
Nat Biotechnol. 2015 Jul;33(7):694-6. doi: 10.1038/nbt.3274.
Nat Biotechnol. 2015.
PMID: 26154005
No abstract available.
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Design and synthesis of dihydrobenzofuran amides as orally bioavailable, centrally active γ-secretase modulators.
Pettersson M, Johnson DS, Subramanyam C, Bales KR, am Ende CW, Fish BA, Green ME, Kauffman GW, Lira R, Mullins PB, Navaratnam T, Sakya SM, Stiff CM, Tran TP, Vetelino BC, Xie L, Zhang L, Pustilnik LR, Wood KM, O'Donnell CJ.
Pettersson M, et al. Among authors: navaratnam t.
Bioorg Med Chem Lett. 2012 Apr 15;22(8):2906-11. doi: 10.1016/j.bmcl.2012.02.059. Epub 2012 Mar 1.
Bioorg Med Chem Lett. 2012.
PMID: 22429469
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Design, synthesis, and pharmacological evaluation of a novel series of pyridopyrazine-1,6-dione γ-secretase modulators.
Pettersson M, Johnson DS, Subramanyam C, Bales KR, am Ende CW, Fish BA, Green ME, Kauffman GW, Mullins PB, Navaratnam T, Sakya SM, Stiff CM, Tran TP, Xie L, Zhang L, Pustilnik LR, Vetelino BC, Wood KM, Pozdnyakov N, Verhoest PR, O'Donnell CJ.
Pettersson M, et al. Among authors: navaratnam t.
J Med Chem. 2014 Feb 13;57(3):1046-62. doi: 10.1021/jm401782h. Epub 2014 Jan 28.
J Med Chem. 2014.
PMID: 24428186
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Pruritic pigmented papules posing permanent problems. Urticaria pigmentosa (UP) with secondary anetoderma.
Gebauer KA, Navaratnam TE, Holgate C.
Gebauer KA, et al. Among authors: navaratnam te.
Arch Dermatol. 1992 Jan;128(1):107, 110. doi: 10.1001/archderm.128.1.107.
Arch Dermatol. 1992.
PMID: 1739279
No abstract available.
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Bullous pemphigoid and multiple sclerosis.
Gebauer K, Cox J, Gartside J, Navaratnam T.
Gebauer K, et al. Among authors: navaratnam t.
J Am Acad Dermatol. 1990 Aug;23(2 Pt 1):329. doi: 10.1016/s0190-9622(08)81252-2.
J Am Acad Dermatol. 1990.
PMID: 2212136
No abstract available.
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