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Structure-Based Design of an in Vivo Active Selective BRD9 Inhibitor.
J Med Chem. 2016 May 26;59(10):4462-75. doi: 10.1021/acs.jmedchem.5b01865. Epub 2016 Mar 10.
J Med Chem. 2016.
PMID: 26914985
Free PMC article.
Sensitivity and engineered resistance of myeloid leukemia cells to BRD9 inhibition.
Hohmann AF, Martin LJ, Minder JL, Roe JS, Shi J, Steurer S, Bader G, McConnell D, Pearson M, Gerstberger T, Gottschamel T, Thompson D, Suzuki Y, Koegl M, Vakoc CR.
Hohmann AF, et al.
Nat Chem Biol. 2016 Sep;12(9):672-9. doi: 10.1038/nchembio.2115. Epub 2016 Jul 4.
Nat Chem Biol. 2016.
PMID: 27376689
Free PMC article.
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A rationale to target the SWI/SNF complex for cancer therapy.
Hohmann AF, Vakoc CR.
Hohmann AF, et al.
Trends Genet. 2014 Aug;30(8):356-63. doi: 10.1016/j.tig.2014.05.001. Epub 2014 Jun 3.
Trends Genet. 2014.
PMID: 24932742
Free PMC article.
Review.
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BET Bromodomain Inhibition Releases the Mediator Complex from Select cis-Regulatory Elements.
Bhagwat AS, Roe JS, Mok BYL, Hohmann AF, Shi J, Vakoc CR.
Bhagwat AS, et al. Among authors: hohmann af.
Cell Rep. 2016 Apr 19;15(3):519-530. doi: 10.1016/j.celrep.2016.03.054. Epub 2016 Apr 7.
Cell Rep. 2016.
PMID: 27068464
Free PMC article.
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The transcriptional cofactor TRIM33 prevents apoptosis in B lymphoblastic leukemia by deactivating a single enhancer.
Wang E, Kawaoka S, Roe JS, Shi J, Hohmann AF, Xu Y, Bhagwat AS, Suzuki Y, Kinney JB, Vakoc CR.
Wang E, et al. Among authors: hohmann af.
Elife. 2015 Apr 28;4:e06377. doi: 10.7554/eLife.06377.
Elife. 2015.
PMID: 25919951
Free PMC article.
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Rational design of a SOCS1-edited tumor-infiltrating lymphocyte therapy using CRISPR/Cas9 screens.
Schlabach MR, Lin S, Collester ZR, Wrocklage C, Shenker S, Calnan C, Xu T, Gannon HS, Williams LJ, Thompson F, Dunbar PR, LaMothe RA, Garrett TE, Colletti N, Hohmann AF, Tubo NJ, Bullock CP, Le Mercier I, Sofjan K, Merkin JJ, Keegan S, Kryukov GV, Dugopolski C, Stegmeier F, Wong K, Sharp FA, Cadzow L, Benson MJ.
Schlabach MR, et al. Among authors: hohmann af.
J Clin Invest. 2023 Dec 15;133(24):e163096. doi: 10.1172/JCI163096.
J Clin Invest. 2023.
PMID: 38099496
Free PMC article.
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Atrial arrhythmogenicity in aged Scn5a+/DeltaKPQ mice modeling long QT type 3 syndrome and its relationship to Na+ channel expression and cardiac conduction.
Guzadhur L, Pearcey SM, Duehmke RM, Jeevaratnam K, Hohmann AF, Zhang Y, Grace AA, Lei M, Huang CL.
Guzadhur L, et al. Among authors: hohmann af.
Pflugers Arch. 2010 Aug;460(3):593-601. doi: 10.1007/s00424-010-0851-z. Epub 2010 Jun 16.
Pflugers Arch. 2010.
PMID: 20552221
Free PMC article.
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