Davies GJ - Search Results

1

A second-generation ferrocene-iminosugar hybrid with improved fucosidase binding properties.

Hottin A, Scandolera A, Duca L, Wright DW, Davies GJ, Behr JB. Hottin A, et al. Among authors: davies gj. Bioorg Med Chem Lett. 2016 Mar 15;26(6):1546-1549. doi: 10.1016/j.bmcl.2016.02.017. Epub 2016 Feb 9. Bioorg Med Chem Lett. 2016. PMID: 26897594

2

Structural and thermodynamic analyses of α-L-fucosidase inhibitors.

Lammerts van Bueren A, Popat SD, Lin CH, Davies GJ. Lammerts van Bueren A, et al. Among authors: davies gj. Chembiochem. 2010 Sep 24;11(14):1971-4. doi: 10.1002/cbic.201000339. Chembiochem. 2010. PMID: 20665773 No abstract available.

3

α-L-fucosidase inhibition by pyrrolidine-ferrocene hybrids: rationalization of ligand-binding properties by structural studies.

Hottin A, Wright DW, Steenackers A, Delannoy P, Dubar F, Biot C, Davies GJ, Behr JB. Hottin A, et al. Among authors: davies gj. Chemistry. 2013 Jul 15;19(29):9526-33. doi: 10.1002/chem.201301001. Epub 2013 Jun 5. Chemistry. 2013. PMID: 23740878

4

Three dimensional structure of a bacterial α-l-fucosidase with a 5-membered iminocyclitol inhibitor.

Wright DW, Moreno-Vargas AJ, Carmona AT, Robina I, Davies GJ. Wright DW, et al. Among authors: davies gj. Bioorg Med Chem. 2013 Aug 15;21(16):4751-4. doi: 10.1016/j.bmc.2013.05.056. Epub 2013 Jun 13. Bioorg Med Chem. 2013. PMID: 23830696

5

Exploiting the hydrophobic terrain in fucosidases with aryl-substituted pyrrolidine iminosugars.

Hottin A, Wright DW, Davies GJ, Behr JB. Hottin A, et al. Among authors: davies gj. Chembiochem. 2015 Jan 19;16(2):277-83. doi: 10.1002/cbic.201402509. Epub 2014 Nov 26. Chembiochem. 2015. PMID: 25427942

6

Exploring the divalent effect in fucosidase inhibition with stereoisomeric pyrrolidine dimers.

Hottin A, Wright DW, Moreno-Clavijo E, Moreno-Vargas AJ, Davies GJ, Behr JB. Hottin A, et al. Among authors: davies gj. Org Biomol Chem. 2016 May 18;14(20):4718-27. doi: 10.1039/c6ob00647g. Org Biomol Chem. 2016. PMID: 27138139

7

In vitro and in vivo comparative and competitive activity-based protein profiling of GH29 α-l-fucosidases.

Jiang J, Kallemeijn WW, Wright DW, van den Nieuwendijk AMCH, Rohde VC, Folch EC, van den Elst H, Florea BI, Scheij S, Donker-Koopman WE, Verhoek M, Li N, Schürmann M, Mink D, Boot RG, Codée JDC, van der Marel GA, Davies GJ, Aerts JMFG, Overkleeft HS. Jiang J, et al. Among authors: davies gj. Chem Sci. 2015 May 1;6(5):2782-false. doi: 10.1039/c4sc03739a. Epub 2015 Feb 9. Chem Sci. 2015. PMID: 29142681 Free PMC article.

8

Synthetic and Crystallographic Insight into Exploiting sp² Hybridization in the Development of α-l-Fucosidase Inhibitors.

Coyle T, Wu L, Debowski AW, Davies GJ, Stubbs KA. Coyle T, et al. Among authors: davies gj. Chembiochem. 2019 Jun 3;20(11):1365-1368. doi: 10.1002/cbic.201800710. Epub 2019 Mar 18. Chembiochem. 2019. PMID: 30663832 Free PMC article.

9

Direct observation of the protonation state of an imino sugar glycosidase inhibitor upon binding.

Varrot A, Tarling CA, Macdonald JM, Stick RV, Zechel DL, Withers SG, Davies GJ. Varrot A, et al. Among authors: davies gj. J Am Chem Soc. 2003 Jun 25;125(25):7496-7. doi: 10.1021/ja034917k. J Am Chem Soc. 2003. PMID: 12812472

10

Iminosugar glycosidase inhibitors: structural and thermodynamic dissection of the binding of isofagomine and 1-deoxynojirimycin to beta-glucosidases.

Zechel DL, Boraston AB, Gloster T, Boraston CM, Macdonald JM, Tilbrook DM, Stick RV, Davies GJ. Zechel DL, et al. Among authors: davies gj. J Am Chem Soc. 2003 Nov 26;125(47):14313-23. doi: 10.1021/ja036833h. J Am Chem Soc. 2003. PMID: 14624580

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