Skip to main page content
U.S. flag

An official website of the United States government

Dot gov

The .gov means it’s official.
Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you’re on a federal government site.

Https

The site is secure.
The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.

Access keys NCBI Homepage MyNCBI Homepage Main Content Main Navigation

Search Page

Filters

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

Search Results

647 results

Filters applied: . Clear all
Results are displayed in a computed author sort order. The Results By Year timeline is not available.
Page 1
Drug design, synthesis, in vitro and in silico evaluation of selective monoaminoxidase B inhibitors based on 3-acetyl-2-dichlorophenyl-5-aryl-2,3-dihydro-1,3,4-oxadiazole chemical scaffold.
Distinto S, Meleddu R, Yanez M, Cirilli R, Bianco G, Sanna ML, Arridu A, Cossu P, Cottiglia F, Faggi C, Ortuso F, Alcaro S, Maccioni E. Distinto S, et al. Among authors: bianco g. Eur J Med Chem. 2016 Jan 27;108:542-552. doi: 10.1016/j.ejmech.2015.12.026. Epub 2015 Dec 17. Eur J Med Chem. 2016. PMID: 26717204
Design, synthesis, and biological evaluation of 1,3-diarylpropenones as dual inhibitors of HIV-1 reverse transcriptase.
Meleddu R, Cannas V, Distinto S, Sarais G, Del Vecchio C, Esposito F, Bianco G, Corona A, Cottiglia F, Alcaro S, Parolin C, Artese A, Scalise D, Fresta M, Arridu A, Ortuso F, Maccioni E, Tramontano E. Meleddu R, et al. Among authors: bianco g. ChemMedChem. 2014 Aug;9(8):1869-79. doi: 10.1002/cmdc.201402015. Epub 2014 May 21. ChemMedChem. 2014. PMID: 24850787
(3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro-1H-indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase.
Meleddu R, Distinto S, Corona A, Bianco G, Cannas V, Esposito F, Artese A, Alcaro S, Matyus P, Bogdan D, Cottiglia F, Tramontano E, Maccioni E. Meleddu R, et al. Among authors: bianco g. Eur J Med Chem. 2015 Mar 26;93:452-60. doi: 10.1016/j.ejmech.2015.02.032. Epub 2015 Feb 20. Eur J Med Chem. 2015. PMID: 25728026
Isatin: a privileged scaffold for the design of carbonic anhydrase inhibitors.
Melis C, Meleddu R, Angeli A, Distinto S, Bianco G, Capasso C, Cottiglia F, Angius R, Supuran CT, Maccioni E. Melis C, et al. Among authors: bianco g. J Enzyme Inhib Med Chem. 2017 Dec;32(1):68-73. doi: 10.1080/14756366.2016.1235042. Epub 2016 Oct 24. J Enzyme Inhib Med Chem. 2017. PMID: 27775452 Free PMC article.
N-Acylbenzenesulfonamide Dihydro-1,3,4-oxadiazole Hybrids: Seeking Selectivity toward Carbonic Anhydrase Isoforms.
Bianco G, Meleddu R, Distinto S, Cottiglia F, Gaspari M, Melis C, Corona A, Angius R, Angeli A, Taverna D, Alcaro S, Leitans J, Kazaks A, Tars K, Supuran CT, Maccioni E. Bianco G, et al. ACS Med Chem Lett. 2017 Jun 21;8(8):792-796. doi: 10.1021/acsmedchemlett.7b00205. eCollection 2017 Aug 10. ACS Med Chem Lett. 2017. PMID: 28835790 Free PMC article.
Targeting Tumor Associated Carbonic Anhydrases IX and XII: Highly Isozyme Selective Coumarin and Psoralen Inhibitors.
Melis C, Distinto S, Bianco G, Meleddu R, Cottiglia F, Fois B, Taverna D, Angius R, Alcaro S, Ortuso F, Gaspari M, Angeli A, Del Prete S, Capasso C, Supuran CT, Maccioni E. Melis C, et al. Among authors: bianco g. ACS Med Chem Lett. 2018 Jun 6;9(7):725-729. doi: 10.1021/acsmedchemlett.8b00170. eCollection 2018 Jul 12. ACS Med Chem Lett. 2018. PMID: 30034608 Free PMC article.
Isatin thiazoline hybrids as dual inhibitors of HIV-1 reverse transcriptase.
Meleddu R, Distinto S, Corona A, Tramontano E, Bianco G, Melis C, Cottiglia F, Maccioni E. Meleddu R, et al. Among authors: bianco g. J Enzyme Inhib Med Chem. 2017 Dec;32(1):130-136. doi: 10.1080/14756366.2016.1238366. Epub 2016 Oct 21. J Enzyme Inhib Med Chem. 2017. PMID: 27766892 Free PMC article.
647 results