Novellino E - Search Results

1

Structure-based drug design targeting the cell membrane receptor GPBAR1: exploiting the bile acid scaffold towards selective agonism.

Di Leva FS, Festa C, Renga B, Sepe V, Novellino E, Fiorucci S, Zampella A, Limongelli V. Di Leva FS, et al. Among authors: novellino e. Sci Rep. 2015 Nov 16;5:16605. doi: 10.1038/srep16605. Sci Rep. 2015. PMID: 26567894 Free PMC article.

2

Synthesis, pharmacological evaluation, and molecular modeling studies of novel peptidic CAAX analogues as farnesyl-protein-transferase inhibitors.

Santagada V, Caliendo G, Severino B, Lavecchia A, Perissutti E, Fiorino F, Zampella A, Sepe V, Califano D, Santelli G, Novellino E. Santagada V, et al. Among authors: novellino e. J Med Chem. 2006 Mar 23;49(6):1882-90. doi: 10.1021/jm0506165. J Med Chem. 2006. PMID: 16539374

3

Modeling of Cdc25B dual specifity protein phosphatase inhibitors: docking of ligands and enzymatic inhibition mechanism.

Lavecchia A, Cosconati S, Limongelli V, Novellino E. Lavecchia A, et al. Among authors: novellino e. ChemMedChem. 2006 May;1(5):540-50. doi: 10.1002/cmdc.200500092. ChemMedChem. 2006. PMID: 16892390

4

Ensemble-docking approach on BACE-1: pharmacophore perception and guidelines for drug design.

Limongelli V, Marinelli L, Cosconati S, Braun HA, Schmidt B, Novellino E. Limongelli V, et al. Among authors: novellino e. ChemMedChem. 2007 May;2(5):667-78. doi: 10.1002/cmdc.200600314. ChemMedChem. 2007. PMID: 17407105

5

Homology modeling of NR2B modulatory domain of NMDA receptor and analysis of ifenprodil binding.

Marinelli L, Cosconati S, Steinbrecher T, Limongelli V, Bertamino A, Novellino E, Case DA. Marinelli L, et al. Among authors: novellino e. ChemMedChem. 2007 Oct;2(10):1498-510. doi: 10.1002/cmdc.200700091. ChemMedChem. 2007. PMID: 17849398

6

Acetic acid aldose reductase inhibitors bearing a five-membered heterocyclic core with potent topical activity in a visual impairment rat model.

La Motta C, Sartini S, Salerno S, Simorini F, Taliani S, Marini AM, Da Settimo F, Marinelli L, Limongelli V, Novellino E. La Motta C, et al. Among authors: novellino e. J Med Chem. 2008 Jun 12;51(11):3182-93. doi: 10.1021/jm701613h. Epub 2008 May 2. J Med Chem. 2008. PMID: 18452283

7

Ethyl 8-fluoro-6-(3-nitrophenyl)-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate as novel, highly potent, and safe antianxiety agent.

Anzini M, Braile C, Valenti S, Cappelli A, Vomero S, Marinelli L, Limongelli V, Novellino E, Betti L, Giannaccini G, Lucacchini A, Ghelardini C, Norcini M, Makovec F, Giorgi G, Ian Fryer R. Anzini M, et al. Among authors: novellino e. J Med Chem. 2008 Aug 14;51(15):4730-43. doi: 10.1021/jm8002944. Epub 2008 Jul 19. J Med Chem. 2008. PMID: 18637672

8

Design, synthesis, and biological evaluation of novel aminobisphosphonates possessing an in vivo antitumor activity through a gammadelta-T lymphocytes-mediated activation mechanism.

Simoni D, Gebbia N, Invidiata FP, Eleopra M, Marchetti P, Rondanin R, Baruchello R, Provera S, Marchioro C, Tolomeo M, Marinelli L, Limongelli V, Novellino E, Kwaasi A, Dunford J, Buccheri S, Caccamo N, Dieli F. Simoni D, et al. Among authors: novellino e. J Med Chem. 2008 Nov 13;51(21):6800-7. doi: 10.1021/jm801003y. Epub 2008 Oct 21. J Med Chem. 2008. PMID: 18937434

9

Breaking the dogma of the metal-coordinating carboxylate group in integrin ligands: introducing hydroxamic acids to the MIDAS to tune potency and selectivity.

Heckmann D, Laufer B, Marinelli L, Limongelli V, Novellino E, Zahn G, Stragies R, Kessler H. Heckmann D, et al. Among authors: novellino e. Angew Chem Int Ed Engl. 2009;48(24):4436-40. doi: 10.1002/anie.200900206. Angew Chem Int Ed Engl. 2009. PMID: 19343753

10

Membrane charge dependent states of the beta-amyloid fragment Abeta (16-35) with differently charged micelle aggregates.

Grimaldi M, Scrima M, Esposito C, Vitiello G, Ramunno A, Limongelli V, D'Errico G, Novellino E, D'Ursi AM. Grimaldi M, et al. Among authors: novellino e. Biochim Biophys Acta. 2010 Mar;1798(3):660-71. doi: 10.1016/j.bbamem.2009.12.012. Epub 2010 Jan 4. Biochim Biophys Acta. 2010. PMID: 20045392 Free article.

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