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Antileishmanial activity of new thiophene-indole hybrids: Design, synthesis, biological and cytotoxic evaluation, and chemometric studies.
Bioorg Med Chem. 2016 Sep 15;24(18):3972-3977. doi: 10.1016/j.bmc.2016.04.057. Epub 2016 Apr 26.
Bioorg Med Chem. 2016.
PMID: 27515718
Free article.
2-Amino-thiophene derivatives present antileishmanial activity mediated by apoptosis and immunomodulation in vitro.
Rodrigues KA, Dias CN, Néris PL, Rocha Jda C, Scotti MT, Scotti L, Mascarenhas SR, Veras RC, de Medeiros IA, Keesen Tde S, de Oliveira TB, de Lima Mdo C, Balliano TL, de Aquino TM, de Moura RO, Mendonça Junior FJ, de Oliveira MR.
Rodrigues KA, et al. Among authors: neris pl.
Eur J Med Chem. 2015 Dec 1;106:1-14. doi: 10.1016/j.ejmech.2015.10.011. Epub 2015 Oct 17.
Eur J Med Chem. 2015.
PMID: 26513640
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Neolignan Licarin A presents effect against Leishmania (Leishmania) major associated with immunomodulation in vitro.
Néris PL, Caldas JP, Rodrigues YK, Amorim FM, Leite JA, Rodrigues-Mascarenhas S, Barbosa-Filho JM, Rodrigues LC, Oliveira MR.
Néris PL, et al.
Exp Parasitol. 2013 Oct;135(2):307-13. doi: 10.1016/j.exppara.2013.07.007. Epub 2013 Jul 24.
Exp Parasitol. 2013.
PMID: 23891943
Free article.
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Immunomodulatory activity of ouabain in Leishmania leishmania amazonensis-infected Swiss mice.
Jacob PL, Leite JA, Alves AK, Rodrigues YK, Amorim FM, Néris PL, Oliveira MR, Rodrigues-Mascarenhas S.
Jacob PL, et al. Among authors: neris pl.
Parasitol Res. 2013 Mar;112(3):1313-21. doi: 10.1007/s00436-012-3146-9. Epub 2012 Oct 4.
Parasitol Res. 2013.
PMID: 23052777
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Morita-Baylis-Hillman adduct shows in vitro activity against Leishmania (Viannia) braziliensis associated with a reduction in IL-6 and IL-10 but independent of nitric oxide.
Amorim FM, Rodrigues YK, Barbosa TP, Néris PL, Caldas JP, Sousa SC, Leite JA, Rodrigues-Mascarenhas S, Vasconcellos ML, Oliveira MR.
Amorim FM, et al. Among authors: neris pl.
Parasitology. 2013 Jan;140(1):29-38. doi: 10.1017/S0031182012001291. Epub 2012 Aug 20.
Parasitology. 2013.
PMID: 22906971
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Efficient synthesis of 16 aromatic Morita-Baylis-Hillman adducts: Biological evaluation on Leishmania amazonensis and Leishmania chagasi.
Junior CG, de Assis PA, Silva FP, Sousa SC, de Andrade NG, Barbosa TP, Nerís PL, Segundo LV, Anjos IC, Carvalho GA, Rocha GB, Oliveira MR, Vasconcellos ML.
Junior CG, et al. Among authors: neris pl.
Bioorg Chem. 2010 Dec;38(6):279-84. doi: 10.1016/j.bioorg.2010.08.002. Epub 2010 Sep 19.
Bioorg Chem. 2010.
PMID: 20855101
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