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Discovery of 2-[1-(4,4-Difluorocyclohexyl)piperidin-4-yl]-6-fluoro-3-oxo-2,3-dihydro-1H-isoindole-4-carboxamide (NMS-P118): A Potent, Orally Available, and Highly Selective PARP-1 Inhibitor for Cancer Therapy.
Papeo G, Posteri H, Borghi D, Busel AA, Caprera F, Casale E, Ciomei M, Cirla A, Corti E, D'Anello M, Fasolini M, Forte B, Galvani A, Isacchi A, Khvat A, Krasavin MY, Lupi R, Orsini P, Perego R, Pesenti E, Pezzetta D, Rainoldi S, Riccardi-Sirtori F, Scolaro A, Sola F, Zuccotto F, Felder ER, Donati D, Montagnoli A. Papeo G, et al. J Med Chem. 2015 Sep 10;58(17):6875-98. doi: 10.1021/acs.jmedchem.5b00680. Epub 2015 Aug 26. J Med Chem. 2015. PMID: 26222319
A straightforward total synthesis of (-)-chaetominine.
Malgesini B, Forte B, Borghi D, Quartieri F, Gennari C, Papeo G. Malgesini B, et al. Among authors: papeo g. Chemistry. 2009 Aug 10;15(32):7922-7929. doi: 10.1002/chem.200900793. Chemistry. 2009. PMID: 19562787
A submarine journey: the pyrrole-imidazole alkaloids.
Forte B, Malgesini B, Piutti C, Quartieri F, Scolaro A, Papeo G. Forte B, et al. Among authors: papeo g. Mar Drugs. 2009 Nov 27;7(4):705-53. doi: 10.3390/md7040705. Mar Drugs. 2009. PMID: 20098608 Free PMC article. Review.
PARP inhibitors in cancer therapy: an update.
Papeo G, Casale E, Montagnoli A, Cirla A. Papeo G, et al. Expert Opin Ther Pat. 2013 Apr;23(4):503-14. doi: 10.1517/13543776.2013.768615. Epub 2013 Feb 5. Expert Opin Ther Pat. 2013. PMID: 23379721 Review.
Discovery and optimization of pyrrolo[1,2-a]pyrazinones leads to novel and selective inhibitors of PIM kinases.
Casuscelli F, Ardini E, Avanzi N, Casale E, Cervi G, D'Anello M, Donati D, Faiardi D, Ferguson RD, Fogliatto G, Galvani A, Marsiglio A, Mirizzi DG, Montemartini M, Orrenius C, Papeo G, Piutti C, Salom B, Felder ER. Casuscelli F, et al. Among authors: papeo g. Bioorg Med Chem. 2013 Dec 1;21(23):7364-80. doi: 10.1016/j.bmc.2013.09.054. Epub 2013 Oct 2. Bioorg Med Chem. 2013. PMID: 24139169
19 results