Design, synthesis and in vitro evaluation of novel SARS-CoV-2 3CLpro covalent inhibitors.
Stille JK, Tjutrins J, Wang G, Venegas FA, Hennecker C, Rueda AM, Sharon I, Blaine N, Miron CE, Pinus S, Labarre A, Plescia J, Burai Patrascu M, Zhang X, Wahba AS, Vlaho D, Huot MJ, Schmeing TM, Mittermaier AK, Moitessier N.
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Eur J Med Chem. 2022 Feb 5;229:114046. doi: 10.1016/j.ejmech.2021.114046. Epub 2021 Dec 11.
Eur J Med Chem. 2022.
PMID: 34995923
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