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A fast capillary electrophoresis method to assess the binding affinity of recombinant antithrombin toward heparin directly from cell culture supernatants.
J Pharm Biomed Anal. 2015;111:64-70. doi: 10.1016/j.jpba.2015.02.042. Epub 2015 Mar 19.
J Pharm Biomed Anal. 2015.
PMID: 25863018
Antithrombin is not protective against renal ischaemia-reperfusion injury.
Bourti Y, Saller F, Bianchini EP, Pautus S, Duong van Huyen JP, Marie AL, Tran NT, Molina TJ, Taverna M, Lerolle N, Borgel D.
Bourti Y, et al. Among authors: pautus s.
Thromb Haemost. 2017 Jan 26;117(2):422-425. doi: 10.1160/TH16-06-0451. Epub 2016 Oct 27.
Thromb Haemost. 2017.
PMID: 27786339
No abstract available.
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Characterization of the Annonaceous acetogenin, annonacinone, a natural product inhibitor of plasminogen activator inhibitor-1.
Pautus S, Alami M, Adam F, Bernadat G, Lawrence DA, De Carvalho A, Ferry G, Rupin A, Hamze A, Champy P, Bonneau N, Gloanec P, Peglion JL, Brion JD, Bianchini EP, Borgel D.
Pautus S, et al.
Sci Rep. 2016 Nov 23;6:36462. doi: 10.1038/srep36462.
Sci Rep. 2016.
PMID: 27876785
Free PMC article.
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New 7-methylguanine derivatives targeting the influenza polymerase PB2 cap-binding domain.
Pautus S, Sehr P, Lewis J, Fortuné A, Wolkerstorfer A, Szolar O, Guilligay D, Lunardi T, Décout JL, Cusack S.
Pautus S, et al.
J Med Chem. 2013 Nov 14;56(21):8915-30. doi: 10.1021/jm401369y. Epub 2013 Nov 6.
J Med Chem. 2013.
PMID: 24134208
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Synthesis and CYP26A1 inhibitory activity of 1-[benzofuran-2-yl-(4-alkyl/aryl-phenyl)-methyl]-1H-triazoles.
Pautus S, Yee SW, Jayne M, Coogan MP, Simons C.
Pautus S, et al.
Bioorg Med Chem. 2006 Jun 1;14(11):3643-53. doi: 10.1016/j.bmc.2006.01.018. Epub 2006 Feb 3.
Bioorg Med Chem. 2006.
PMID: 16458519
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Design and synthesis of substituted imidazole and triazole N-phenylbenzo[d]oxazolamine inhibitors of retinoic acid metabolizing enzyme CYP26.
Pautus S, Aboraia AS, Bassett CE, Brancale A, Coogan MP, Simons C.
Pautus S, et al.
J Enzyme Inhib Med Chem. 2009 Apr;24(2):487-98. doi: 10.1080/14756360802218334.
J Enzyme Inhib Med Chem. 2009.
PMID: 18608743
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