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First evidence that oligopyridines, α-helix foldamers, inhibit Mcl-1 and sensitize ovarian carcinoma cells to Bcl-xL-targeting strategies.
J Med Chem. 2015 Feb 26;58(4):1644-68. doi: 10.1021/jm500672y. Epub 2015 Feb 4.
J Med Chem. 2015.
PMID: 25585174
Structural characterizations of oligopyridyl foldamers, α-helix mimetics.
Santos JS, Voisin-Chiret AS, Burzicki G, Sebaoun L, Sebban M, Lohier JF, Legay R, Oulyadi H, Bureau R, Rault S.
Santos JS, et al. Among authors: burzicki g.
J Chem Inf Model. 2012 Feb 27;52(2):429-39. doi: 10.1021/ci200424a. Epub 2012 Jan 17.
J Chem Inf Model. 2012.
PMID: 22196240
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