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Selective inhibitors of the FK506-binding protein 51 by induced fit.
Nat Chem Biol. 2015 Jan;11(1):33-7. doi: 10.1038/nchembio.1699. Epub 2014 Dec 1.
Nat Chem Biol. 2015.
PMID: 25436518
Pharmacological Inhibition of the Psychiatric Risk Factor FKBP51 Has Anxiolytic Properties.
Hartmann J, Wagner KV, Gaali S, Kirschner A, Kozany C, Rühter G, Dedic N, Häusl AS, Hoeijmakers L, Westerholz S, Namendorf C, Gerlach T, Uhr M, Chen A, Deussing JM, Holsboer F, Hausch F, Schmidt MV.
Hartmann J, et al. Among authors: ruhter g.
J Neurosci. 2015 Jun 17;35(24):9007-16. doi: 10.1523/JNEUROSCI.4024-14.2015.
J Neurosci. 2015.
PMID: 26085626
Free PMC article.
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Identification of Atuveciclib (BAY 1143572), the First Highly Selective, Clinical PTEFb/CDK9 Inhibitor for the Treatment of Cancer.
Lücking U, Scholz A, Lienau P, Siemeister G, Kosemund D, Bohlmann R, Briem H, Terebesi I, Meyer K, Prelle K, Denner K, Bömer U, Schäfer M, Eis K, Valencia R, Ince S, von Nussbaum F, Mumberg D, Ziegelbauer K, Klebl B, Choidas A, Nussbaumer P, Baumann M, Schultz-Fademrecht C, Rühter G, Eickhoff J, Brands M.
Lücking U, et al. Among authors: ruhter g.
ChemMedChem. 2017 Nov 8;12(21):1776-1793. doi: 10.1002/cmdc.201700447. Epub 2017 Oct 16.
ChemMedChem. 2017.
PMID: 28961375
Free PMC article.
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Spirocyclic nonpeptide glycoprotein IIb-IIIa antagonists. Part 3: synthesis and SAR of potent and specific 2,8-diazaspiro[4.5]decanes.
Mehrotra MM, Heath JA, Rose JW, Smyth MS, Seroogy J, Volkots DL, Ruhter G, Schotten T, Alaimo L, Park G, Pandey A, Scarborough RM.
Mehrotra MM, et al. Among authors: ruhter g.
Bioorg Med Chem Lett. 2002 Apr 8;12(7):1103-7. doi: 10.1016/s0960-894x(02)00095-1.
Bioorg Med Chem Lett. 2002.
PMID: 11909727
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Spirocyclic nonpeptide glycoprotein IIb-IIIa antagonists. Part 2: design of potent antagonists containing the 3-azaspiro[5.5]undecanes.
Pandey A, Seroogy J, Volkots D, Smyth MS, Rose J, Mehrotra MM, Heath J, Ruhter G, Schotten T, Scarborough RM.
Pandey A, et al. Among authors: ruhter g.
Bioorg Med Chem Lett. 2001 May 21;11(10):1293-6. doi: 10.1016/s0960-894x(01)00216-5.
Bioorg Med Chem Lett. 2001.
PMID: 11392540
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Spirocyclic nonpeptide glycoprotein IIb-IIIa antagonists. Part 1: design of potent and specific 3,9-diazaspiro[5.5]undecanes.
Smyth MS, Rose J, Mehrotra MM, Heath J, Ruhter G, Schotten T, Seroogy J, Volkots D, Pandey A, Scarborough RM.
Smyth MS, et al. Among authors: ruhter g.
Bioorg Med Chem Lett. 2001 May 21;11(10):1289-92. doi: 10.1016/s0960-894x(01)00215-3.
Bioorg Med Chem Lett. 2001.
PMID: 11392539
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Fused bicyclic Gly-Asp beta-turn mimics with potent affinity for GPIIb-IIIa. Exploration of the arginine isostere.
Fisher MJ, Giese U, Harms CS, Kinnick MD, Lindstrom TD, McCowan JR, Mest HJ, Morin JM Jr, Mullaney JT, Paal M, Rapp A, Rühter G, Ruterbories KJ, Sall DJ, Scarborough RM, Schotten T, Stenzel W, Towner RD, Um SL, Utterback BG, Wyss VL, Jakubowski JA.
Fisher MJ, et al. Among authors: ruhter g.
Bioorg Med Chem Lett. 2000 Feb 21;10(4):385-9. doi: 10.1016/s0960-894x(00)00008-1.
Bioorg Med Chem Lett. 2000.
PMID: 10714506
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Fused bicyclic Gly-Asp beta-turn mimics with specific affinity for GPIIb-IIIa.
Fisher MJ, Arfstan AE, Giese U, Gunn BP, Harms CS, Khau V, Kinnick MD, Lindstrom TD, Martinelli MJ, Mest HJ, Mohr M, Morin JM Jr, Mullaney JT, Nunes A, Paal M, Rapp A, Rühter G, Ruterbories KJ, Sall DJ, Scarborough RM, Schotten T, Sommer B, Stenzel W, Towner RD, Um SL, et al.
Fisher MJ, et al. Among authors: ruhter g.
J Med Chem. 1999 Nov 18;42(23):4875-89. doi: 10.1021/jm990365y.
J Med Chem. 1999.
PMID: 10579850
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