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A cell-permeable inhibitor to trap Gαq proteins in the empty pocket conformation.
Chem Biol. 2014 Jul 17;21(7):890-902. doi: 10.1016/j.chembiol.2014.06.003.
Chem Biol. 2014.
PMID: 25036778
Free PMC article.
A small-molecule inhibitor of Nipah virus envelope protein-mediated membrane fusion.
Niedermeier S, Singethan K, Rohrer SG, Matz M, Kossner M, Diederich S, Maisner A, Schmitz J, Hiltensperger G, Baumann K, Holzgrabe U, Schneider-Schaulies J.
Niedermeier S, et al. Among authors: hiltensperger g.
J Med Chem. 2009 Jul 23;52(14):4257-65. doi: 10.1021/jm900411s.
J Med Chem. 2009.
PMID: 19499921
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Synthesis and structure-activity relationships of new quinolone-type molecules against Trypanosoma brucei.
Hiltensperger G, Jones NG, Niedermeier S, Stich A, Kaiser M, Jung J, Puhl S, Damme A, Braunschweig H, Meinel L, Engstler M, Holzgrabe U.
Hiltensperger G, et al.
J Med Chem. 2012 Mar 22;55(6):2538-48. doi: 10.1021/jm101439s. Epub 2012 Mar 12.
J Med Chem. 2012.
PMID: 22376072
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N-(3-Cyanophenyl)-2-phenylacetamide, an effective inhibitor of morbillivirus-induced membrane fusion with low cytotoxicity.
Singethan K, Hiltensperger G, Kendl S, Wohlfahrt J, Plattet P, Holzgrabe U, Schneider-Schaulies J.
Singethan K, et al. Among authors: hiltensperger g.
J Gen Virol. 2010 Nov;91(Pt 11):2762-72. doi: 10.1099/vir.0.025650-0. Epub 2010 Aug 4.
J Gen Virol. 2010.
PMID: 20685931
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Quinolone Amides as Antitrypanosomal Lead Compounds with In Vivo Activity.
Hiltensperger G, Hecht N, Kaiser M, Rybak JC, Hoerst A, Dannenbauer N, Müller-Buschbaum K, Bruhn H, Esch H, Lehmann L, Meinel L, Holzgrabe U.
Hiltensperger G, et al.
Antimicrob Agents Chemother. 2016 Jul 22;60(8):4442-52. doi: 10.1128/AAC.01757-15. Print 2016 Aug.
Antimicrob Agents Chemother. 2016.
PMID: 27139467
Free PMC article.
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Mechanism for active membrane fusion triggering by morbillivirus attachment protein.
Ader N, Brindley M, Avila M, Örvell C, Horvat B, Hiltensperger G, Schneider-Schaulies J, Vandevelde M, Zurbriggen A, Plemper RK, Plattet P.
Ader N, et al. Among authors: hiltensperger g.
J Virol. 2013 Jan;87(1):314-26. doi: 10.1128/JVI.01826-12. Epub 2012 Oct 17.
J Virol. 2013.
PMID: 23077316
Free PMC article.
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