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Structural and biological exploration of phe(3)-phe(4)-modified endomorphin-2 peptidomimetics.
ACS Med Chem Lett. 2013 Jul 11;4(8):795-9. doi: 10.1021/ml400189r. eCollection 2013 Aug 8.
ACS Med Chem Lett. 2013.
PMID: 24900748
Free PMC article.
Synthesis, pharmacological evaluation and conformational investigation of endomorphin-2 hybrid analogues.
Lesma G, Salvadori S, Airaghi F, Bojnik E, Borsodi A, Recca T, Sacchetti A, Balboni G, Silvani A.
Lesma G, et al. Among authors: airaghi f.
Mol Divers. 2013 Feb;17(1):19-31. doi: 10.1007/s11030-012-9399-5. Epub 2012 Nov 4.
Mol Divers. 2013.
PMID: 23124951
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The diketopiperazine-fused tetrahydro-β-carboline scaffold as a model peptidomimetic with an unusual α-turn secondary structure.
Airaghi F, Fiorati A, Lesma G, Musolino M, Sacchetti A, Silvani A.
Airaghi F, et al.
Beilstein J Org Chem. 2013;9:147-54. doi: 10.3762/bjoc.9.17. Epub 2013 Jan 22.
Beilstein J Org Chem. 2013.
PMID: 23399789
Free PMC article.
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3-Oxo-hexahydro-1H-isoindole-4-carboxylic Acid as a Drug Chiral Bicyclic Scaffold: Structure-Based Design and Preparation of Conformationally Constrained Covalent and Noncovalent Prolyl Oligopeptidase Inhibitors.
Mariaule G, De Cesco S, Airaghi F, Kurian J, Schiavini P, Rocheleau S, Huskić I, Auclair K, Mittermaier A, Moitessier N.
Mariaule G, et al. Among authors: airaghi f.
J Med Chem. 2016 May 12;59(9):4221-34. doi: 10.1021/acs.jmedchem.5b01296. Epub 2015 Dec 14.
J Med Chem. 2016.
PMID: 26619267
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An experimental procedure to perform mechanical characterization of small-sized bone specimens from thin femoral cortical wall.
Gastaldi D, Baleani M, Fognani R, Airaghi F, Bonanni L, Vena P.
Gastaldi D, et al. Among authors: airaghi f.
J Mech Behav Biomed Mater. 2020 Dec;112:104046. doi: 10.1016/j.jmbbm.2020.104046. Epub 2020 Sep 1.
J Mech Behav Biomed Mater. 2020.
PMID: 32911224
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