Godessart N - Search Results

1

Discovery of LAS101057: A Potent, Selective, and Orally Efficacious A2B Adenosine Receptor Antagonist.

Eastwood P, Esteve C, González J, Fonquerna S, Aiguadé J, Carranco I, Doménech T, Aparici M, Miralpeix M, Albertí J, Córdoba M, Fernández R, Pont M, Godessart N, Prats N, Loza MI, Cadavid MI, Nueda A, Vidal B. Eastwood P, et al. Among authors: godessart n. ACS Med Chem Lett. 2010 Dec 20;2(3):213-8. doi: 10.1021/ml100249e. eCollection 2011 Mar 10. ACS Med Chem Lett. 2010. PMID: 24900298 Free PMC article.

2

Discovery and characterization of 4'-(2-furyl)-N-pyridin-3-yl-4,5'-bipyrimidin-2'-amine (LAS38096), a potent, selective, and efficacious A2B adenosine receptor antagonist.

Vidal B, Nueda A, Esteve C, Domenech T, Benito S, Reinoso RF, Pont M, Calbet M, López R, Cadavid MI, Loza MI, Cárdenas A, Godessart N, Beleta J, Warrellow G, Ryder H. Vidal B, et al. Among authors: godessart n. J Med Chem. 2007 May 31;50(11):2732-6. doi: 10.1021/jm061333v. Epub 2007 May 1. J Med Chem. 2007. PMID: 17469811

3

Design, synthesis, and structure-activity relationships of aminopyridine N-oxides, a novel scaffold for the potent and selective inhibition of p38 mitogen activated protein kinase.

Lumeras W, Caturla F, Vidal L, Esteve C, Balagué C, Orellana A, Domínguez M, Roca R, Huerta JM, Godessart N, Vidal B. Lumeras W, et al. Among authors: godessart n. J Med Chem. 2009 Sep 10;52(17):5531-45. doi: 10.1021/jm9008604. J Med Chem. 2009. PMID: 19678708

4

Discovery of a novel class of zwitterionic, potent, selective and orally active S1P₁ direct agonists.

Aguilar N, Mir M, Grima PM, López M, Segarra V, Esteban L, Moreno I, Godessart N, Tarrasón G, Domenech T, Vilella D, Armengol C, Córdoba M, Sabaté M, Casals D, Domínguez M. Aguilar N, et al. Among authors: godessart n. Bioorg Med Chem Lett. 2012 Dec 15;22(24):7672-6. doi: 10.1016/j.bmcl.2012.09.110. Epub 2012 Oct 11. Bioorg Med Chem Lett. 2012. PMID: 23141913

5

Profiling of dihydroorotate dehydrogenase, p38 and JAK inhibitors in the rat adjuvant-induced arthritis model: a translational study.

Balagué C, Pont M, Prats N, Godessart N. Balagué C, et al. Among authors: godessart n. Br J Pharmacol. 2012 Jun;166(4):1320-32. doi: 10.1111/j.1476-5381.2012.01836.x. Br J Pharmacol. 2012. PMID: 22229697 Free PMC article.

6

Phosphodiesterase 7A1 is expressed in human CD4+ naïve T cells at higher levels than in CD4+ memory cells and is not required during their CD3/CD28-dependent activation.

Nueda A, García-Roger N, Domenech T, Godessart N, Cárdenas A, Santamaría-Babi LF, Beleta J. Nueda A, et al. Among authors: godessart n. Cell Immunol. 2006 Jul;242(1):31-8. doi: 10.1016/j.cellimm.2006.09.001. Epub 2006 Oct 10. Cell Immunol. 2006. PMID: 17034773

7

The sphingosine-1-phosphate receptor-1 antagonist, W146, causes early and short-lasting peripheral blood lymphopenia in mice.

Tarrasón G, Aulí M, Mustafa S, Dolgachev V, Domènech MT, Prats N, Domínguez M, López R, Aguilar N, Calbet M, Pont M, Milligan G, Kunkel SL, Godessart N. Tarrasón G, et al. Among authors: godessart n. Int Immunopharmacol. 2011 Nov;11(11):1773-9. doi: 10.1016/j.intimp.2011.07.004. Epub 2011 Jul 26. Int Immunopharmacol. 2011. PMID: 21798372

8

Prediction of the skin permeability of topical drugs using in silico and in vitro models.

Alonso C, Carrer V, Espinosa S, Zanuy M, Córdoba M, Vidal B, Domínguez M, Godessart N, Coderch L, Pont M. Alonso C, et al. Among authors: godessart n. Eur J Pharm Sci. 2019 Aug 1;136:104945. doi: 10.1016/j.ejps.2019.05.023. Epub 2019 Jun 1. Eur J Pharm Sci. 2019. PMID: 31163216

9

Synthesis and biological evaluation of 3,4-diaryloxazolones: A new class of orally active cyclooxygenase-2 inhibitors.

Puig C, Crespo MI, Godessart N, Feixas J, Ibarzo J, Jiménez JM, Soca L, Cardelús I, Heredia A, Miralpeix M, Puig J, Beleta J, Huerta JM, López M, Segarra V, Ryder H, Palacios JM. Puig C, et al. Among authors: godessart n. J Med Chem. 2000 Jan 27;43(2):214-23. doi: 10.1021/jm991106b. J Med Chem. 2000. PMID: 10649977

10

Pharmacological blockade of CCR1 ameliorates murine arthritis and alters cytokine networks in vivo.

Amat M, Benjamim CF, Williams LM, Prats N, Terricabras E, Beleta J, Kunkel SL, Godessart N. Amat M, et al. Among authors: godessart n. Br J Pharmacol. 2006 Nov;149(6):666-75. doi: 10.1038/sj.bjp.0706912. Epub 2006 Oct 3. Br J Pharmacol. 2006. PMID: 17016504 Free PMC article.

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