Creation of Customized Bioactivity within a 14-Membered Macrolide Scaffold: Design, Synthesis, and Biological Evaluation Using a Family-18 Chitinase.
Sugawara A, Maita N, Gouda H, Yamamoto T, Hirose T, Kimura S, Saito Y, Nakano H, Kasai T, Nakano H, Shiomi K, Hirono S, Watanabe T, Taniguchi H, Omura S, Sunazuka T.
Sugawara A, et al. Among authors: shiomi k.
J Med Chem. 2015 Jun 25;58(12):4984-97. doi: 10.1021/acs.jmedchem.5b00175. Epub 2015 Jun 12.
J Med Chem. 2015.
PMID: 26030312