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Glucocorticoid receptor modulators informed by crystallography lead to a new rationale for receptor selectivity, function, and implications for structure-based design.
J Med Chem. 2014 Feb 13;57(3):849-60. doi: 10.1021/jm401616g. Epub 2014 Feb 4.
J Med Chem. 2014.
PMID: 24446728
Indole Glucocorticoid Receptor Antagonists Active in a Model of Dyslipidemia Act via a Unique Association with an Agonist Binding Site.
Luz JG, Carson MW, Condon B, Clawson D, Pustilnik A, Kohlman DT, Barr RJ, Bean JS, Dill MJ, Sindelar DK, Maletic M, Coghlan MJ.
Luz JG, et al. Among authors: kohlman dt.
J Med Chem. 2015 Aug 27;58(16):6607-18. doi: 10.1021/acs.jmedchem.5b00736. Epub 2015 Aug 7.
J Med Chem. 2015.
PMID: 26218343
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Structure-activity relationships of SERMs optimized for uterine antagonism and ovarian safety.
Richardson TI, Frank SA, Wang M, Clarke CA, Jones SA, Ying BP, Kohlman DT, Wallace OB, Shepherd TA, Dally RD, Palkowitz AD, Geiser AG, Bryant HU, Henck JW, Cohen IR, Rudmann DG, McCann DJ, Coutant DE, Oldham SW, Hummel CW, Fong KC, Hinklin R, Lewis G, Tian H, Dodge JA.
Richardson TI, et al. Among authors: kohlman dt.
Bioorg Med Chem Lett. 2007 Jul 1;17(13):3544-9. doi: 10.1016/j.bmcl.2007.04.044. Epub 2007 Apr 24.
Bioorg Med Chem Lett. 2007.
PMID: 17482463
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Discovery of selective N-[3-(1-methyl-piperidine-4-carbonyl)-phenyl]-benzamide-based 5-HT₁ F receptor agonists: Evolution from bicyclic to monocyclic cores.
Zhang D, Blanco MJ, Ying BP, Kohlman D, Liang SX, Victor F, Chen Q, Krushinski J, Filla SA, Hudziak KJ, Mathes BM, Cohen MP, Zacherl D, Nelson DL, Wainscott DB, Nutter SE, Gough WH, Schaus JM, Xu YC.
Zhang D, et al.
Bioorg Med Chem Lett. 2015 Oct 1;25(19):4337-41. doi: 10.1016/j.bmcl.2015.07.042. Epub 2015 Jul 22.
Bioorg Med Chem Lett. 2015.
PMID: 26271587
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Design, synthesis and evaluation of bicyclic benzamides as novel 5-HT1F receptor agonists.
Zhang D, Kohlman D, Krushinski J, Liang S, Ying BP, Reilly JE, Dinn SR, Wainscott DB, Nutter S, Gough W, Nelson DL, Schaus JM, Xu YC.
Zhang D, et al.
Bioorg Med Chem Lett. 2004 Dec 20;14(24):6011-6. doi: 10.1016/j.bmcl.2004.09.079.
Bioorg Med Chem Lett. 2004.
PMID: 15546719
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N-Methyl-5-tert-butyltryptamine: A novel, highly potent 5-HT1D receptor agonist.
Xu YC, Schaus JM, Walker C, Krushinski J, Adham N, Zgombick JM, Liang SX, Kohlman DT, Audia JE.
Xu YC, et al. Among authors: kohlman dt.
J Med Chem. 1999 Feb 11;42(3):526-31. doi: 10.1021/jm9805945.
J Med Chem. 1999.
PMID: 9986723
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Oxidative C-C bond-forming reaction of electron-rich alkylbenzyl ether with trimethylvinyloxysilane.
Ying BP, Trogden BG, Kohlman DT, Liang SX, Xu YC.
Ying BP, et al. Among authors: kohlman dt.
Org Lett. 2004 May 13;6(10):1523-6. doi: 10.1021/ol036314j.
Org Lett. 2004.
PMID: 15128226
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