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Allosteric modulators of human A2B adenosine receptor.
Trincavelli ML, Giacomelli C, Daniele S, Taliani S, Cosimelli B, Laneri S, Severi E, Barresi E, Pugliesi I, Greco G, Novellino E, Da Settimo F, Martini C. Trincavelli ML, et al. Among authors: pugliesi i. Biochim Biophys Acta. 2014 Mar;1840(3):1194-203. doi: 10.1016/j.bbagen.2013.12.021. Epub 2013 Dec 19. Biochim Biophys Acta. 2014. PMID: 24361612
Derivatives of benzimidazol-2-ylquinoline and benzimidazol-2-ylisoquinoline as selective A1 adenosine receptor antagonists with stimulant activity on human colon motility.
Cosimelli B, Taliani S, Greco G, Novellino E, Sala A, Severi E, Da Settimo F, La Motta C, Pugliesi I, Antonioli L, Fornai M, Colucci R, Blandizzi C, Daniele S, Trincavelli ML, Martini C. Cosimelli B, et al. Among authors: pugliesi i. ChemMedChem. 2011 Oct 4;6(10):1909-18. doi: 10.1002/cmdc.201100284. Epub 2011 Jul 27. ChemMedChem. 2011. PMID: 21796795
3-aryl-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-one: a novel template for the design of highly selective A₂B adenosine receptor antagonists.
Taliani S, Pugliesi I, Barresi E, Simorini F, Salerno S, La Motta C, Marini AM, Cosimelli B, Cosconati S, Di Maro S, Marinelli L, Daniele S, Trincavelli ML, Greco G, Novellino E, Martini C, Da Settimo F. Taliani S, et al. Among authors: pugliesi i. J Med Chem. 2012 Feb 23;55(4):1490-9. doi: 10.1021/jm201177b. Epub 2012 Feb 7. J Med Chem. 2012. PMID: 22257095
Modulation of A2B adenosine receptor by 1-Benzyl-3-ketoindole derivatives.
Taliani S, Trincavelli ML, Cosimelli B, Laneri S, Severi E, Barresi E, Pugliesi I, Daniele S, Giacomelli C, Greco G, Novellino E, Martini C, Da Settimo F. Taliani S, et al. Among authors: pugliesi i. Eur J Med Chem. 2013 Nov;69:331-7. doi: 10.1016/j.ejmech.2013.09.001. Epub 2013 Sep 8. Eur J Med Chem. 2013. PMID: 24077183
Modulation of PAR(1) signalling by benzimidazole compounds.
Asteriti S, Daniele S, Porchia F, Dell'Anno MT, Fazzini A, Pugliesi I, Trincavelli ML, Taliani S, Martini C, Mazzoni MR, Gilchrist A. Asteriti S, et al. Among authors: pugliesi i. Br J Pharmacol. 2012 Sep;167(1):80-94. doi: 10.1111/j.1476-5381.2012.01974.x. Br J Pharmacol. 2012. PMID: 22519452 Free PMC article.
A3 receptor ligands: past, present and future trends.
Taliani S, Pugliesi I, Bellandi M, La Motta C, Da Settimo F. Taliani S, et al. Among authors: pugliesi i. Curr Top Med Chem. 2010;10(10):942-75. doi: 10.2174/156802610791293109. Curr Top Med Chem. 2010. PMID: 20370658 Review.
3-(Fur-2-yl)-10-(2-phenylethyl)-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-one, a novel adenosine receptor antagonist with A(2A)-mediated neuroprotective effects.
Scatena A, Fornai F, Trincavelli ML, Taliani S, Daniele S, Pugliesi I, Cosconati S, Martini C, Da Settimo F. Scatena A, et al. Among authors: pugliesi i. ACS Chem Neurosci. 2011 Sep 21;2(9):526-35. doi: 10.1021/cn200036s. Epub 2011 Jun 10. ACS Chem Neurosci. 2011. PMID: 22860174 Free PMC article.
34 results