Prisinzano TE - Search Results

1

Development of functionally selective, small molecule agonists at kappa opioid receptors.

Zhou L, Lovell KM, Frankowski KJ, Slauson SR, Phillips AM, Streicher JM, Stahl E, Schmid CL, Hodder P, Madoux F, Cameron MD, Prisinzano TE, Aubé J, Bohn LM. Zhou L, et al. Among authors: prisinzano te. J Biol Chem. 2013 Dec 20;288(51):36703-16. doi: 10.1074/jbc.M113.504381. Epub 2013 Nov 1. J Biol Chem. 2013. PMID: 24187130 Free PMC article.

2

A MOR Antagonist with High Potency and Antagonist Efficacy among Diastereomeric C9-Alkyl-Substituted N-Phenethyl-5-(3-hydroxy)phenylmorphans.

Chambers DR, Sulima A, Luo D, Prisinzano TE, Jacobson AE, Rice KC. Chambers DR, et al. Among authors: prisinzano te. Molecules. 2023 Jul 14;28(14):5411. doi: 10.3390/molecules28145411. Molecules. 2023. PMID: 37513283 Free PMC article.

3

An opioid agonist that does not induce mu-opioid receptor--arrestin interactions or receptor internalization.

Groer CE, Tidgewell K, Moyer RA, Harding WW, Rothman RB, Prisinzano TE, Bohn LM. Groer CE, et al. Among authors: prisinzano te. Mol Pharmacol. 2007 Feb;71(2):549-57. doi: 10.1124/mol.106.028258. Epub 2006 Nov 7. Mol Pharmacol. 2007. PMID: 17090705 Free PMC article.

4

A comparison of noninternalizing (herkinorin) and internalizing (DAMGO) mu-opioid agonists on cellular markers related to opioid tolerance and dependence.

Xu H, Partilla JS, Wang X, Rutherford JM, Tidgewell K, Prisinzano TE, Bohn LM, Rothman RB. Xu H, et al. Among authors: prisinzano te. Synapse. 2007 Mar;61(3):166-75. doi: 10.1002/syn.20356. Synapse. 2007. PMID: 17152090

5

Herkinorin analogues with differential beta-arrestin-2 interactions.

Tidgewell K, Groer CE, Harding WW, Lozama A, Schmidt M, Marquam A, Hiemstra J, Partilla JS, Dersch CM, Rothman RB, Bohn LM, Prisinzano TE. Tidgewell K, et al. Among authors: prisinzano te. J Med Chem. 2008 Apr 24;51(8):2421-31. doi: 10.1021/jm701162g. Epub 2008 Apr 2. J Med Chem. 2008. PMID: 18380425 Free PMC article.

6

Synthetic studies of neoclerodane diterpenes from Salvia divinorum: role of the furan in affinity for opioid receptors.

Simpson DS, Lovell KM, Lozama A, Han N, Day VW, Dersch CM, Rothman RB, Prisinzano TE. Simpson DS, et al. Among authors: prisinzano te. Org Biomol Chem. 2009 Sep 21;7(18):3748-56. doi: 10.1039/b905148a. Epub 2009 Jul 14. Org Biomol Chem. 2009. PMID: 19707679 Free PMC article.

7

Fragment-based screening by X-ray crystallography, MS and isothermal titration calorimetry to identify PNMT (phenylethanolamine N-methyltransferase) inhibitors.

Drinkwater N, Vu H, Lovell KM, Criscione KR, Collins BM, Prisinzano TE, Poulsen SA, McLeish MJ, Grunewald GL, Martin JL. Drinkwater N, et al. Among authors: prisinzano te. Biochem J. 2010 Oct 1;431(1):51-61. doi: 10.1042/BJ20100651. Biochem J. 2010. PMID: 20642456

8

Utilizing nature as a source of new probes for opioid pharmacology.

Lovell KM, Simpson DS, Cunningham CW, Prisinzano TE. Lovell KM, et al. Among authors: prisinzano te. Future Med Chem. 2009 May;1(2):285-301. doi: 10.4155/fmc.09.22. Future Med Chem. 2009. PMID: 21425970 Review.

9

Synthesis of neoclerodane diterpenes and their pharmacological effects.

Lovell KM, Prevatt-Smith KM, Lozama A, Prisinzano TE. Lovell KM, et al. Among authors: prisinzano te. Top Curr Chem. 2011;299:141-85. doi: 10.1007/128_2010_82. Top Curr Chem. 2011. PMID: 21630517 Review.

10

Antinociceptive effects of herkinorin, a MOP receptor agonist derived from salvinorin A in the formalin test in rats: new concepts in mu opioid receptor pharmacology: from a symposium on new concepts in mu-opioid pharmacology.

Lamb K, Tidgewell K, Simpson DS, Bohn LM, Prisinzano TE. Lamb K, et al. Among authors: prisinzano te. Drug Alcohol Depend. 2012 Mar 1;121(3):181-8. doi: 10.1016/j.drugalcdep.2011.10.026. Epub 2011 Nov 26. Drug Alcohol Depend. 2012. PMID: 22119134 Free PMC article.

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