Rami M - Search Results

1

Hypoxia-targeting carbonic anhydrase IX inhibitors by a new series of nitroimidazole-sulfonamides/sulfamides/sulfamates.

Rami M, Dubois L, Parvathaneni NK, Alterio V, van Kuijk SJ, Monti SM, Lambin P, De Simone G, Supuran CT, Winum JY. Rami M, et al. J Med Chem. 2013 Nov 14;56(21):8512-20. doi: 10.1021/jm4009532. Epub 2013 Oct 31. J Med Chem. 2013. PMID: 24128000

2

Carbonic anhydrase IX: a new druggable target for the design of antitumor agents.

Winum JY, Rami M, Scozzafava A, Montero JL, Supuran C. Winum JY, et al. Among authors: rami m. Med Res Rev. 2008 May;28(3):445-63. doi: 10.1002/med.20112. Med Res Rev. 2008. PMID: 17880011 Review.

3

Carbonic anhydrase inhibitors: copper(II) complexes of polyamino-polycarboxylamido aromatic/heterocyclic sulfonamides are very potent inhibitors of the tumor-associated isoforms IX and XII.

Rami M, Winum JY, Innocenti A, Montero JL, Scozzafava A, Supuran CT. Rami M, et al. Bioorg Med Chem Lett. 2008 Jan 15;18(2):836-41. doi: 10.1016/j.bmcl.2007.11.025. Epub 2007 Nov 13. Bioorg Med Chem Lett. 2008. PMID: 18042384

4

Carbonic anhydrase inhibitors: design of membrane-impermeant copper(II) complexes of DTPA-, DOTA-, and TETA-tailed sulfonamides targeting the tumor-associated transmembrane isoform IX.

Rami M, Cecchi A, Montero JL, Innocenti A, Vullo D, Scozzafava A, Winum JY, Supuran CT. Rami M, et al. ChemMedChem. 2008 Nov;3(11):1780-8. doi: 10.1002/cmdc.200800267. ChemMedChem. 2008. PMID: 18956406

5

Carbonic anhydrase inhibitor coated gold nanoparticles selectively inhibit the tumor-associated isoform IX over the cytosolic isozymes I and II.

Stiti M, Cecchi A, Rami M, Abdaoui M, Barragan-Montero V, Scozzafava A, Guari Y, Winum JY, Supuran CT. Stiti M, et al. Among authors: rami m. J Am Chem Soc. 2008 Dec 3;130(48):16130-1. doi: 10.1021/ja805558k. J Am Chem Soc. 2008. PMID: 18989963

6

Carbonic anhydrase inhibitors: 2-substituted-1,3,4-thiadiazole-5-sulfamides act as powerful and selective inhibitors of the mitochondrial isozymes VA and VB over the cytosolic and membrane-associated carbonic anhydrases I, II and IV.

Smaine FZ, Pacchiano F, Rami M, Barragan-Montero V, Vullo D, Scozzafava A, Winum JY, Supuran CT. Smaine FZ, et al. Among authors: rami m. Bioorg Med Chem Lett. 2008 Dec 15;18(24):6332-5. doi: 10.1016/j.bmcl.2008.10.093. Epub 2008 Nov 1. Bioorg Med Chem Lett. 2008. PMID: 18990571

7

Sulfonamides incorporating boroxazolidone moieties are potent inhibitors of the transmembrane, tumor-associated carbonic anhydrase isoforms IX and XII.

Rami M, Maresca A, Smaine FZ, Montero JL, Scozzafava A, Winum JY, Supuran CT. Rami M, et al. Bioorg Med Chem Lett. 2011 May 15;21(10):2975-9. doi: 10.1016/j.bmcl.2011.03.055. Epub 2011 Mar 21. Bioorg Med Chem Lett. 2011. PMID: 21470859

8

Synthesis of rhodamine B-benzenesulfonamide conjugates and their inhibitory activity against human α- and bacterial/fungal β-carbonic anhydrases.

Rami M, Innocenti A, Montero JL, Scozzafava A, Winum JY, Supuran CT. Rami M, et al. Bioorg Med Chem Lett. 2011 Sep 15;21(18):5210-3. doi: 10.1016/j.bmcl.2011.07.045. Epub 2011 Jul 21. Bioorg Med Chem Lett. 2011. PMID: 21821413

9

(Hetero)aryl substituted thiazol-2,4-yl scaffold as human carbonic anhydrase I, II, VII and XIV activators.

Rami M, Winum JY, Supuran CT, Melnyk P, Yous S. Rami M, et al. J Enzyme Inhib Med Chem. 2019 Dec;34(1):224-229. doi: 10.1080/14756366.2018.1543292. J Enzyme Inhib Med Chem. 2019. PMID: 30734616 Free PMC article.

10

Targeting carbonic anhydrase IX by nitroimidazole based sulfamides enhances the therapeutic effect of tumor irradiation: a new concept of dual targeting drugs.

Dubois L, Peeters SG, van Kuijk SJ, Yaromina A, Lieuwes NG, Saraya R, Biemans R, Rami M, Parvathaneni NK, Vullo D, Vooijs M, Supuran CT, Winum JY, Lambin P. Dubois L, et al. Among authors: rami m. Radiother Oncol. 2013 Sep;108(3):523-8. doi: 10.1016/j.radonc.2013.06.018. Epub 2013 Jul 9. Radiother Oncol. 2013. PMID: 23849171 Free article.

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