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Optimization of pyrrolamides as mycobacterial GyrB ATPase inhibitors: structure-activity relationship and in vivo efficacy in a mouse model of tuberculosis.
Antimicrob Agents Chemother. 2014;58(1):61-70. doi: 10.1128/AAC.01751-13. Epub 2013 Oct 14.
Antimicrob Agents Chemother. 2014.
PMID: 24126580
Free PMC article.
Novel N-linked aminopiperidine-based gyrase inhibitors with improved hERG and in vivo efficacy against Mycobacterium tuberculosis.
Hameed P S, Patil V, Solapure S, Sharma U, Madhavapeddi P, Raichurkar A, Chinnapattu M, Manjrekar P, Shanbhag G, Puttur J, Shinde V, Menasinakai S, Rudrapatana S, Achar V, Awasthy D, Nandishaiah R, Humnabadkar V, Ghosh A, Narayan C, Ramya VK, Kaur P, Sharma S, Werngren J, Hoffner S, Panduga V, Kumar CN, Reddy J, Kumar K N M, Ganguly S, Bharath S, Bheemarao U, Mukherjee K, Arora U, Gaonkar S, Coulson M, Waterson D, Sambandamurthy VK, de Sousa SM.
Hameed P S, et al. Among authors: chinnapattu m.
J Med Chem. 2014 Jun 12;57(11):4889-905. doi: 10.1021/jm500432n. Epub 2014 May 23.
J Med Chem. 2014.
PMID: 24809953
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Aminoazabenzimidazoles, a novel class of orally active antimalarial agents.
Hameed P S, Chinnapattu M, Shanbag G, Manjrekar P, Koushik K, Raichurkar A, Patil V, Jatheendranath S, Rudrapatna SS, Barde SP, Rautela N, Awasthy D, Morayya S, Narayan C, Kavanagh S, Saralaya R, Bharath S, Viswanath P, Mukherjee K, Bandodkar B, Srivastava A, Panduga V, Reddy J, Prabhakar KR, Sinha A, Jiménez-Díaz MB, Martínez MS, Angulo-Barturen I, Ferrer S, Sanz LM, Gamo FJ, Duffy S, Avery VM, Magistrado PA, Lukens AK, Wirth DF, Waterson D, Balasubramanian V, Iyer PS, Narayanan S, Hosagrahara V, Sambandamurthy VK, Ramachandran S.
Hameed P S, et al. Among authors: chinnapattu m.
J Med Chem. 2014 Jul 10;57(13):5702-13. doi: 10.1021/jm500535j. Epub 2014 Jun 24.
J Med Chem. 2014.
PMID: 24914738
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UDP-N-acetylmuramic acid l-alanine ligase (MurC) inhibition in a tolC mutant Escherichia coli strain leads to cell death.
Humnabadkar V, Prabhakar KR, Narayan A, Sharma S, Guptha S, Manjrekar P, Chinnapattu M, Ramachandran V, Hameed SP, Ravishankar S, Chatterji M.
Humnabadkar V, et al. Among authors: chinnapattu m.
Antimicrob Agents Chemother. 2014 Oct;58(10):6165-71. doi: 10.1128/AAC.02890-14. Epub 2014 Aug 11.
Antimicrob Agents Chemother. 2014.
PMID: 25114134
Free PMC article.
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Left-Hand Side Exploration of Novel Bacterial Topoisomerase Inhibitors to Improve Selectivity against hERG Binding.
Hameed P S, Manjrekar P, Raichurkar A, Shinde V, Puttur J, Shanbhag G, Chinnapattu M, Patil V, Rudrapatana S, Sharma S, Kumar CN, Nandishaiah R, Madhavapeddi P, Sriram D, Solapure S, Sambandamurthy VK.
Hameed P S, et al. Among authors: chinnapattu m.
ACS Med Chem Lett. 2015 May 22;6(7):741-6. doi: 10.1021/ml500531p. eCollection 2015 Jul 9.
ACS Med Chem Lett. 2015.
PMID: 26191359
Free PMC article.
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Pyrazolopyrimidines establish MurC as a vulnerable target in Pseudomonas aeruginosa and Escherichia coli.
Hameed P S, Manjrekar P, Chinnapattu M, Humnabadkar V, Shanbhag G, Kedari C, Mudugal NV, Ambady A, de Jonge BL, Sadler C, Paul B, Sriram S, Kaur P, Guptha S, Raichurkar A, Fleming P, Eyermann CJ, McKinney DC, Sambandamurthy VK, Panda M, Ravishankar S.
Hameed P S, et al. Among authors: chinnapattu m.
ACS Chem Biol. 2014 Oct 17;9(10):2274-82. doi: 10.1021/cb500360c. Epub 2014 Aug 5.
ACS Chem Biol. 2014.
PMID: 25035921
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Synthesis and biological evaluation of adamantane-based aminophenols as a novel class of antiplasmodial agents.
Chinnapattu M, Sathiyanarayanan KI, Iyer PS.
Chinnapattu M, et al.
Bioorg Med Chem Lett. 2015 Feb 15;25(4):952-5. doi: 10.1016/j.bmcl.2014.12.037. Epub 2014 Dec 19.
Bioorg Med Chem Lett. 2015.
PMID: 25599834
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Validation of an enantioselective LC-MS/MS method to quantify enantiomers of (±)-OTX015 in mice plasma: Lack of in vivo inversion of (-)-OTX015 to its antipode.
Balaji N, Chinnapattu M, Dixit A, Sahu P, P S S, Mullangi R.
Balaji N, et al. Among authors: chinnapattu m.
Biomed Chromatogr. 2017 Apr;31(4). doi: 10.1002/bmc.3853. Epub 2016 Oct 14.
Biomed Chromatogr. 2017.
PMID: 27632936
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