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Structure-based design, parallel synthesis, structure-activity relationship, and molecular modeling studies of thiocarbamates, new potent non-nucleoside HIV-1 reverse transcriptase inhibitor isosteres of phenethylthiazolylthiourea derivatives.
Ranise A, Spallarossa A, Cesarini S, Bondavalli F, Schenone S, Bruno O, Menozzi G, Fossa P, Mosti L, La Colla M, Sanna G, Murreddu M, Collu G, Busonera B, Marongiu ME, Pani A, La Colla P, Loddo R. Ranise A, et al. J Med Chem. 2005 Jun 2;48(11):3858-73. doi: 10.1021/jm049252r. J Med Chem. 2005. PMID: 15916438
Assuming as a lead compound O-[2-(phthalimido)ethyl]phenylthiocarbamate 12, one of the precursors of the previously described acylthiocarbamates (Ranise, A.; et al. ...The lead optimization strategy led to para-substituted TCs 31, 33, 34, 39, 40, 41, 44, 45, …
Assuming as a lead compound O-[2-(phthalimido)ethyl]phenylthiocarbamate 12, one of the precursors of the previously described acylthi …
Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 1: Parallel synthesis, molecular modelling and structure-activity relationship studies on O-[2-(hetero)arylethyl]-N-phenylthiocarbamates.
Cesarini S, Spallarossa A, Ranise A, Fossa P, La Colla P, Sanna G, Collu G, Loddo R. Cesarini S, et al. Among authors: ranise a. Bioorg Med Chem. 2008 Apr 1;16(7):4160-72. doi: 10.1016/j.bmc.2007.12.050. Epub 2007 Dec 25. Bioorg Med Chem. 2008. PMID: 18226532
Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 2: Parallel synthesis, molecular modelling and structure-activity relationship studies on analogues of O-(2-phenylethyl)-N-phenylthiocarbamate.
Cesarini S, Spallarossa A, Ranise A, Bruno O, La Colla P, Secci B, Collu G, Loddo R. Cesarini S, et al. Among authors: ranise a. Bioorg Med Chem. 2008 Apr 1;16(7):4173-85. doi: 10.1016/j.bmc.2007.12.046. Epub 2007 Dec 25. Bioorg Med Chem. 2008. PMID: 18226533
Parallel one-pot synthesis and structure-activity relationship study of symmetric formimidoester disulfides as a novel class of potent non-nucleoside HIV-1 reverse transcriptase inhibitors.
Cesarini S, Spallarossa A, Ranise A, Schenone S, Bruno O, La Colla P, Casula L, Collu G, Sanna G, Loddo R. Cesarini S, et al. Among authors: ranise a. Bioorg Med Chem. 2008 Jun 15;16(12):6353-63. doi: 10.1016/j.bmc.2008.05.010. Epub 2008 May 7. Bioorg Med Chem. 2008. PMID: 18502646
Parallel synthesis, molecular modelling and further structure-activity relationship studies of new acylthiocarbamates as potent non-nucleoside HIV-1 reverse transcriptase inhibitors.
Spallarossa A, Cesarini S, Ranise A, Schenone S, Bruno O, Borassi A, La Colla P, Pezzullo M, Sanna G, Collu G, Secci B, Loddo R. Spallarossa A, et al. Among authors: ranise a. Eur J Med Chem. 2009 May;44(5):2190-201. doi: 10.1016/j.ejmech.2008.10.032. Epub 2008 Nov 5. Eur J Med Chem. 2009. PMID: 19058881
6-amino-4-oxo-1,3-diphenyl-2-thioxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl derivatives as a new class of potent inhibitors of Interleukin-8-induced neutrophil chemotaxis.
Cesarini S, Spallarossa A, Ranise A, Bruno O, Arduino N, Bertolotto M, Dallegri F, Tognolini M, Gobbetti T, Barocelli E. Cesarini S, et al. Among authors: ranise a. Bioorg Med Chem. 2009 May 15;17(10):3580-7. doi: 10.1016/j.bmc.2009.04.006. Epub 2009 Apr 11. Bioorg Med Chem. 2009. PMID: 19394230
108 results