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Cell-permeable stapled peptides based on HIV-1 integrase inhibitors derived from HIV-1 gene products.
Nomura W, Aikawa H, Ohashi N, Urano E, Métifiot M, Fujino M, Maddali K, Ozaki T, Nozue A, Narumi T, Hashimoto C, Tanaka T, Pommier Y, Yamamoto N, Komano JA, Murakami T, Tamamura H. Nomura W, et al. Among authors: hashimoto c. ACS Chem Biol. 2013 Oct 18;8(10):2235-44. doi: 10.1021/cb400495h. Epub 2013 Aug 15. ACS Chem Biol. 2013. PMID: 23898787 Free PMC article.
Peptide HIV-1 integrase inhibitors from HIV-1 gene products.
Suzuki S, Urano E, Hashimoto C, Tsutsumi H, Nakahara T, Tanaka T, Nakanishi Y, Maddali K, Han Y, Hamatake M, Miyauchi K, Pommier Y, Beutler JA, Sugiura W, Fuji H, Hoshino T, Itotani K, Nomura W, Narumi T, Yamamoto N, Komano JA, Tamamura H. Suzuki S, et al. Among authors: hashimoto c. J Med Chem. 2010 Jul 22;53(14):5356-60. doi: 10.1021/jm1003528. J Med Chem. 2010. PMID: 20586421 Free PMC article.
Peptidic HIV integrase inhibitors derived from HIV gene products: structure-activity relationship studies.
Suzuki S, Maddali K, Hashimoto C, Urano E, Ohashi N, Tanaka T, Ozaki T, Arai H, Tsutsumi H, Narumi T, Nomura W, Yamamoto N, Pommier Y, Komano JA, Tamamura H. Suzuki S, et al. Among authors: hashimoto c. Bioorg Med Chem. 2010 Sep 15;18(18):6771-5. doi: 10.1016/j.bmc.2010.07.050. Epub 2010 Jul 25. Bioorg Med Chem. 2010. PMID: 20708407 Free PMC article.
Evaluation of a synthetic C34 trimer of HIV-1 gp41 as AIDS vaccines.
Hashimoto C, Nomura W, Ohya A, Urano E, Miyauchi K, Narumi T, Aikawa H, Komano JA, Yamamoto N, Tamamura H. Hashimoto C, et al. Bioorg Med Chem. 2012 May 15;20(10):3287-91. doi: 10.1016/j.bmc.2012.03.050. Epub 2012 Mar 29. Bioorg Med Chem. 2012. PMID: 22507207
Multimerized CHR-derived peptides as HIV-1 fusion inhibitors.
Nomura W, Hashimoto C, Suzuki T, Ohashi N, Fujino M, Murakami T, Yamamoto N, Tamamura H. Nomura W, et al. Among authors: hashimoto c. Bioorg Med Chem. 2013 Aug 1;21(15):4452-8. doi: 10.1016/j.bmc.2013.05.060. Epub 2013 Jun 5. Bioorg Med Chem. 2013. PMID: 23800723 Free article.
CXCR4-derived synthetic peptides inducing anti-HIV-1 antibodies.
Hashimoto C, Nomura W, Narumi T, Fujino M, Nakahara T, Yamamoto N, Murakami T, Tamamura H. Hashimoto C, et al. Bioorg Med Chem. 2013 Nov 15;21(22):6878-85. doi: 10.1016/j.bmc.2013.09.037. Epub 2013 Sep 21. Bioorg Med Chem. 2013. PMID: 24119449
313 results