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Carbonic anhydrase inhibitors. Phenols incorporating 2- or 3-pyridyl-ethenylcarbonyl and tertiary amine moieties strongly inhibit Saccharomyces cerevisiae β-carbonic anhydrase.
J Enzyme Inhib Med Chem. 2014 Aug;29(4):495-9. doi: 10.3109/14756366.2013.806497. Epub 2013 Jul 1.
J Enzyme Inhib Med Chem. 2014.
PMID: 23808805
A magnificent enzyme superfamily: carbonic anhydrases, their purification and characterization.
Ozensoy Guler O, Capasso C, Supuran CT.
Ozensoy Guler O, et al.
J Enzyme Inhib Med Chem. 2016 Oct;31(5):689-94. doi: 10.3109/14756366.2015.1059333. Epub 2015 Jun 29.
J Enzyme Inhib Med Chem. 2016.
PMID: 26118417
Review.
Item in Clipboard
Carbonic anhydrase IX as a novel candidate in liquid biopsy.
Ozensoy Guler O, Supuran CT, Capasso C.
Ozensoy Guler O, et al.
J Enzyme Inhib Med Chem. 2020 Dec;35(1):255-260. doi: 10.1080/14756366.2019.1697251.
J Enzyme Inhib Med Chem. 2020.
PMID: 31790601
Free PMC article.
Review.
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Is carbonic anhydrase inhibition useful as a complementary therapy of Covid-19 infection?
Deniz S, Uysal TK, Capasso C, Supuran CT, Ozensoy Guler O.
Deniz S, et al. Among authors: ozensoy guler o.
J Enzyme Inhib Med Chem. 2021 Dec;36(1):1230-1235. doi: 10.1080/14756366.2021.1924165.
J Enzyme Inhib Med Chem. 2021.
PMID: 34074197
Free PMC article.
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The inhibitory effect of boric acid on hypoxia-regulated tumour-associated carbonic anhydrase IX.
Yusuf ZS, Uysal TK, Simsek E, Nocentini A, Osman SM, Supuran CT, Özensoy Güler Ö.
Yusuf ZS, et al. Among authors: ozensoy guler o.
J Enzyme Inhib Med Chem. 2022 Dec;37(1):1340-1345. doi: 10.1080/14756366.2022.2072837.
J Enzyme Inhib Med Chem. 2022.
PMID: 35535546
Free PMC article.
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Differential in vitro inhibitory effects of anticancer drugs on tumor-associated carbonic anhydrase isozymes CA IX and CA XII.
Ozensoy Guler O, Arslan O, Kockar F.
Ozensoy Guler O, et al.
Methods Find Exp Clin Pharmacol. 2008 Jun;30(5):335-40. doi: 10.1358/mf.2008.30.5.1143022.
Methods Find Exp Clin Pharmacol. 2008.
PMID: 18806891
Free article.
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