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Discovery of a novel pharmacological and structural class of gamma secretase modulators derived from the extract of Actaea racemosa.
ACS Chem Neurosci. 2012 Nov 21;3(11):941-51. doi: 10.1021/cn3000857. Epub 2012 Aug 28.
ACS Chem Neurosci. 2012.
PMID: 23205187
Free PMC article.
Optimization of a natural product-based class of γ-secretase modulators.
Hubbs JL, Fuller NO, Austin WF, Shen R, Creaser SP, McKee TD, Loureiro RM, Tate B, Xia W, Ives J, Bronk BS.
Hubbs JL, et al. Among authors: austin wf.
J Med Chem. 2012 Nov 8;55(21):9270-82. doi: 10.1021/jm300976b. Epub 2012 Oct 15.
J Med Chem. 2012.
PMID: 23030762
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Initial Optimization of a New Series of γ-Secretase Modulators Derived from a Triterpene Glycoside.
Fuller NO, Hubbs JL, Austin WF, Creaser SP, McKee TD, Loureiro RM, Tate B, Xia W, Ives JL, Findeis MA, Bronk BS.
Fuller NO, et al. Among authors: austin wf.
ACS Med Chem Lett. 2012 Aug 29;3(11):908-13. doi: 10.1021/ml300256p. eCollection 2012 Nov 8.
ACS Med Chem Lett. 2012.
PMID: 24900406
Free PMC article.
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Modulation of gamma-secretase for the treatment of Alzheimer's disease.
Tate B, McKee TD, Loureiro RM, Dumin JA, Xia W, Pojasek K, Austin WF, Fuller NO, Hubbs JL, Shen R, Jonker J, Ives J, Bronk BS.
Tate B, et al. Among authors: austin wf.
Int J Alzheimers Dis. 2012;2012:210756. doi: 10.1155/2012/210756. Epub 2012 Dec 19.
Int J Alzheimers Dis. 2012.
PMID: 23320246
Free PMC article.
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Efficacy of SPI-1865, a novel gamma-secretase modulator, in multiple rodent models.
Loureiro RM, Dumin JA, McKee TD, Austin WF, Fuller NO, Hubbs JL, Shen R, Jonker J, Ives J, Bronk BS, Tate B.
Loureiro RM, et al. Among authors: austin wf.
Alzheimers Res Ther. 2013 Apr 18;5(2):19. doi: 10.1186/alzrt173. eCollection 2013.
Alzheimers Res Ther. 2013.
PMID: 23597079
Free PMC article.
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Minimization of drug-drug interaction risk and candidate selection in a natural product-based class of gamma-secretase modulators.
Hubbs JL, Fuller NO, Austin WF, Shen R, Ma J, Gong Z, Li J, McKee TD, Loureiro RM, Tate B, Dumin JA, Ives J, Bronk BS.
Hubbs JL, et al. Among authors: austin wf.
Bioorg Med Chem Lett. 2015 Apr 1;25(7):1621-6. doi: 10.1016/j.bmcl.2015.01.051. Epub 2015 Feb 10.
Bioorg Med Chem Lett. 2015.
PMID: 25708617
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Reactions of (trialkylsilyl)vinylketenes with lithium ynolates: a new benzannulation strategy.
Austin WF, Zhang Y, Danheiser RL.
Austin WF, et al.
Org Lett. 2005 Sep 1;7(18):3905-8. doi: 10.1021/ol051307b.
Org Lett. 2005.
PMID: 16119928
Free PMC article.
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A benzannulation strategy for the synthesis of phenols and heteroaromatic compounds based on the reaction of (trialkylsilyl)vinylketenes with lithium ynolates.
Austin WF, Zhang Y, Danheiser RL.
Austin WF, et al.
Tetrahedron. 2008 Jan 28;64(5):915-925. doi: 10.1016/j.tet.2007.10.113.
Tetrahedron. 2008.
PMID: 19180173
Free PMC article.
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