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Azo-reductase activated budesodine prodrugs for colon targeting.
Bioorg Med Chem Lett. 2012 Dec 15;22(24):7573-7. doi: 10.1016/j.bmcl.2012.10.006. Epub 2012 Oct 17.
Bioorg Med Chem Lett. 2012.
PMID: 23122819
A nitrophenyl-based prodrug type for colorectal targeting of prednisolone, budesonide and celecoxib.
Marquez Ruiz JF, Kedziora K, Pigott M, Keogh B, Windle H, Gavin J, Kelleher DP, Gilmer JF.
Marquez Ruiz JF, et al.
Bioorg Med Chem Lett. 2013 Mar 15;23(6):1693-8. doi: 10.1016/j.bmcl.2013.01.060. Epub 2013 Feb 8.
Bioorg Med Chem Lett. 2013.
PMID: 23416011
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