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New aminoimidazoles as β-secretase (BACE-1) inhibitors showing amyloid-β (Aβ) lowering in brain.
J Med Chem. 2012 Nov 8;55(21):9297-311. doi: 10.1021/jm300991n. Epub 2012 Oct 3.
J Med Chem. 2012.
PMID: 23017051
Core refinement toward permeable β-secretase (BACE-1) inhibitors with low hERG activity.
Ginman T, Viklund J, Malmström J, Blid J, Emond R, Forsblom R, Johansson A, Kers A, Lake F, Sehgelmeble F, Sterky KJ, Bergh M, Lindgren A, Johansson P, Jeppsson F, Fälting J, Gravenfors Y, Rahm F.
Ginman T, et al. Among authors: gravenfors y.
J Med Chem. 2013 Jun 13;56(11):4181-205. doi: 10.1021/jm3011349. Epub 2013 May 20.
J Med Chem. 2013.
PMID: 23126626
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Creation of Novel Cores for β-Secretase (BACE-1) Inhibitors: A Multiparameter Lead Generation Strategy.
Viklund J, Kolmodin K, Nordvall G, Swahn BM, Svensson M, Gravenfors Y, Rahm F.
Viklund J, et al. Among authors: gravenfors y.
ACS Med Chem Lett. 2014 Feb 3;5(4):440-5. doi: 10.1021/ml5000433. eCollection 2014 Apr 10.
ACS Med Chem Lett. 2014.
PMID: 24900855
Free PMC article.
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Discovery of novel pyrrolopyridazine scaffolds as transient receptor potential vanilloid (TRPV1) antagonists.
Dorange I, Forsblom R, Macsari I, Svensson M, Bylund J, Besidski Y, Blid J, Sohn D, Gravenfors Y.
Dorange I, et al. Among authors: gravenfors y.
Bioorg Med Chem Lett. 2012 Nov 15;22(22):6888-95. doi: 10.1016/j.bmcl.2012.09.059. Epub 2012 Sep 25.
Bioorg Med Chem Lett. 2012.
PMID: 23058884
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Phenyl isoxazole voltage-gated sodium channel blockers: structure and activity relationship.
Macsari I, Sandberg L, Besidski Y, Gravenfors Y, Ginman T, Bylund J, Bueters T, Eriksson AB, Lund PE, Venyike E, Arvidsson PI.
Macsari I, et al. Among authors: gravenfors y.
Bioorg Med Chem Lett. 2011 Jul 1;21(13):3871-6. doi: 10.1016/j.bmcl.2011.05.041. Epub 2011 May 18.
Bioorg Med Chem Lett. 2011.
PMID: 21641215
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The Oncolytic Efficacy and in Vivo Pharmacokinetics of [2-(4-Chlorophenyl)quinolin-4-yl](piperidine-2-yl)methanol (Vacquinol-1) Are Governed by Distinct Stereochemical Features.
Hammarström LG, Harmel RK, Granath M, Ringom R, Gravenfors Y, Färnegårdh K, Svensson PH, Wennman D, Lundin G, Roddis Y, Kitambi SS, Bernlind A, Lehmann F, Ernfors P.
Hammarström LG, et al. Among authors: gravenfors y.
J Med Chem. 2016 Sep 22;59(18):8577-92. doi: 10.1021/acs.jmedchem.6b01009. Epub 2016 Sep 8.
J Med Chem. 2016.
PMID: 27607569
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Ultralarge Virtual Screening Identifies SARS-CoV-2 Main Protease Inhibitors with Broad-Spectrum Activity against Coronaviruses.
Luttens A, Gullberg H, Abdurakhmanov E, Vo DD, Akaberi D, Talibov VO, Nekhotiaeva N, Vangeel L, De Jonghe S, Jochmans D, Krambrich J, Tas A, Lundgren B, Gravenfors Y, Craig AJ, Atilaw Y, Sandström A, Moodie LWK, Lundkvist Å, van Hemert MJ, Neyts J, Lennerstrand J, Kihlberg J, Sandberg K, Danielson UH, Carlsson J.
Luttens A, et al. Among authors: gravenfors y.
J Am Chem Soc. 2022 Feb 23;144(7):2905-2920. doi: 10.1021/jacs.1c08402. Epub 2022 Feb 10.
J Am Chem Soc. 2022.
PMID: 35142215
Free PMC article.
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Rapid Construction of a Chloromethyl-Substituted Duocarmycin-like Prodrug.
Bengtsson C, Gravenfors Y.
Bengtsson C, et al. Among authors: gravenfors y.
Molecules. 2023 Jun 16;28(12):4818. doi: 10.3390/molecules28124818.
Molecules. 2023.
PMID: 37375372
Free PMC article.
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