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Design and optimization of quinazoline derivatives as melanin concentrating hormone receptor 1 (MCHR1) antagonists.
Bioorg Med Chem Lett. 2012 May 1;22(9):3157-62. doi: 10.1016/j.bmcl.2012.03.050. Epub 2012 Mar 23.
Bioorg Med Chem Lett. 2012.
PMID: 22487182
Novel pyrazole-3-carboxamide derivatives as cannabinoid-1 (CB1) antagonists: journey from non-polar to polar amides.
Sasmal PK, Reddy DS, Talwar R, Venkatesham B, Balasubrahmanyam D, Kannan M, Srinivas P, Kyasa SK, Devi BN, Jadhav VP, Khan SK, Mohan P, Chaudhury H, Bhuniya D, Iqbal J, Chakrabarti R.
Sasmal PK, et al. Among authors: balasubrahmanyam d.
Bioorg Med Chem Lett. 2011 Jan 1;21(1):562-8. doi: 10.1016/j.bmcl.2010.10.055. Epub 2010 Oct 27.
Bioorg Med Chem Lett. 2011.
PMID: 21075633
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Structure-activity relationship studies of novel pyrazole and imidazole carboxamides as cannabinoid-1 (CB1) antagonists.
Sasmal PK, Talwar R, Swetha J, Balasubrahmanyam D, Venkatesham B, Rawoof KA, Neelima Devi B, Jadhav VP, Khan SK, Mohan P, Srinivasa Reddy D, Nyavanandi VK, Nanduri S, Kyasa SK, Kannan M, Srinivas P, Nadipalli P, Chaudhury H, Sebastian VJ.
Sasmal PK, et al. Among authors: balasubrahmanyam d.
Bioorg Med Chem Lett. 2011 Aug 15;21(16):4913-8. doi: 10.1016/j.bmcl.2011.06.017. Epub 2011 Jul 7.
Bioorg Med Chem Lett. 2011.
PMID: 21741835
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Design and optimization of quinazoline derivatives as melanin concentrating hormone receptor 1 (MCHR1) antagonists: part 2.
Sasmal S, Balasubrahmanyam D, Kanna Reddy HR, Balaji G, Srinivas G, Cheera S, Abbineni C, Sasmal PK, Khanna I, Sebastian VJ, Jadhav VP, Singh MP, Talwar R, Suresh J, Shashikumar D, Harinder Reddy K, Sihorkar V, Frimurer TM, Rist Ø, Elster L, Högberg T.
Sasmal S, et al. Among authors: balasubrahmanyam d.
Bioorg Med Chem Lett. 2012 May 1;22(9):3163-7. doi: 10.1016/j.bmcl.2012.03.049. Epub 2012 Mar 23.
Bioorg Med Chem Lett. 2012.
PMID: 22497763
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