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Cell-based and in-silico studies on the high intrinsic activity of two boron-containing salbutamol derivatives at the human β₂-adrenoceptor.
Bioorg Med Chem. 2012 Jan 15;20(2):933-41. doi: 10.1016/j.bmc.2011.11.054. Epub 2011 Dec 1.
Bioorg Med Chem. 2012.
PMID: 22182578
Function-specific virtual screening for GPCR ligands using a combined scoring method.
Kooistra AJ, Vischer HF, McNaught-Flores D, Leurs R, de Esch IJ, de Graaf C.
Kooistra AJ, et al.
Sci Rep. 2016 Jun 24;6:28288. doi: 10.1038/srep28288.
Sci Rep. 2016.
PMID: 27339552
Free PMC article.
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Non-Imidazole Histamine H₃ Ligands. Part VII. Synthesis, In Vitro and In Vivo Characterization of 5-Substituted-2-thiazol-4-n-propylpiperazines.
Guryn R, Staszewski M, Stasiak A, McNaught Flores D, Fogel WA, Leurs R, Walczyński K.
Guryn R, et al.
Molecules. 2018 Feb 3;23(2):326. doi: 10.3390/molecules23020326.
Molecules. 2018.
PMID: 29401659
Free PMC article.
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4-Hydroxypiperidines and Their Flexible 3-(Amino)propyloxy Analogues as Non-Imidazole Histamine H₃ Receptor Antagonist: Further Structure⁻Activity Relationship Exploration and In Vitro and In Vivo Pharmacological Evaluation.
Olszewska B, Stasiak A, McNaught Flores D, Fogel WA, Leurs R, Walczyński K.
Olszewska B, et al.
Int J Mol Sci. 2018 Apr 19;19(4):1243. doi: 10.3390/ijms19041243.
Int J Mol Sci. 2018.
PMID: 29671795
Free PMC article.
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Design, synthesis, and in vitro and in vivo characterization of 1-{4-[4-(substituted)piperazin-1-yl]butyl}guanidines and their piperidine analogues as histamine H3 receptor antagonists.
Staszewski M, Stasiak A, Karcz T, McNaught Flores D, Fogel WA, Kieć-Kononowicz K, Leurs R, Walczyński K.
Staszewski M, et al.
Medchemcomm. 2019 Jan 11;10(2):234-251. doi: 10.1039/c8md00527c. eCollection 2019 Feb 1.
Medchemcomm. 2019.
PMID: 30881612
Free PMC article.
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Pharmacological Characterization of the Zebrafish (Danio Rerio) Histamine H1 Receptor Reveals the Involvement of the Second Extracellular Loop in the Binding of Histamine.
McNaught-Flores DA, Kooistra AJ, Chen YC, Arias-Montano JA, Panula P, Leurs R.
McNaught-Flores DA, et al.
Mol Pharmacol. 2024 Jan 10;105(2):84-96. doi: 10.1124/molpharm.123.000741.
Mol Pharmacol. 2024.
PMID: 37977823
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Structural and Molecular Determinants for Isoform Bias at Human Histamine H3 Receptor Isoforms.
Rahman SN, McNaught-Flores DA, Huppelschoten Y, da Costa Pereira D, Christopoulos A, Leurs R, Langmead CJ.
Rahman SN, et al. Among authors: mcnaught flores da.
ACS Chem Neurosci. 2023 Feb 15;14(4):645-656. doi: 10.1021/acschemneuro.2c00425. Epub 2023 Jan 26.
ACS Chem Neurosci. 2023.
PMID: 36702158
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