Khalil A - Search Results

1

Synthesis, biological evaluation, and radioiodination of halogenated closo-carboranylthymidine analogues.

Tiwari R, Toppino A, Agarwal HK, Huo T, Byun Y, Gallucci J, Hasabelnaby S, Khalil A, Goudah A, Baiocchi RA, Darby MV, Barth RF, Tjarks W. Tiwari R, et al. Among authors: khalil a. Inorg Chem. 2012 Jan 2;51(1):629-39. doi: 10.1021/ic202150b. Epub 2011 Dec 16. Inorg Chem. 2012. PMID: 22175713 Free PMC article.

2

N3-substituted thymidine bioconjugates for cancer therapy and imaging.

Khalil A, Ishita K, Ali T, Tjarks W. Khalil A, et al. Future Med Chem. 2013 Apr;5(6):677-92. doi: 10.4155/fmc.13.31. Future Med Chem. 2013. PMID: 23617430 Free PMC article. Review.

3

Cellular influx, efflux, and anabolism of 3-carboranyl thymidine analogs: potential boron delivery agents for neutron capture therapy.

Sjuvarsson E, Damaraju VL, Mowles D, Sawyer MB, Tiwari R, Agarwal HK, Khalil A, Hasabelnaby S, Goudah A, Nakkula RJ, Barth RF, Cass CE, Eriksson S, Tjarks W. Sjuvarsson E, et al. Among authors: khalil a. J Pharmacol Exp Ther. 2013 Nov;347(2):388-97. doi: 10.1124/jpet.113.207464. Epub 2013 Sep 4. J Pharmacol Exp Ther. 2013. PMID: 24006340 Free PMC article.

4

Iodine monochloride facilitated deglycosylation, anomerization, and isomerization of 3-substituted thymidine analogues.

Khalil A, Ishita K, Ali T, Tiwari R, Riachy R, Toppino A, Hasabelnaby S, Sayfullin N, Oliver AG, Gallucci J, Huang Z, Tjarks W. Khalil A, et al. Nucleosides Nucleotides Nucleic Acids. 2014;33(12):786-99. doi: 10.1080/15257770.2014.945648. Nucleosides Nucleotides Nucleic Acids. 2014. PMID: 25372994 Free PMC article.

5

Design, synthesis, and biological evaluation of aminothiazole derivatives against the fungal pathogens Histoplasma capsulatum and Cryptococcus neoformans.

Khalil A, Edwards JA, Rappleye CA, Tjarks W. Khalil A, et al. Bioorg Med Chem. 2015 Feb 1;23(3):532-47. doi: 10.1016/j.bmc.2014.12.006. Epub 2014 Dec 10. Bioorg Med Chem. 2015. PMID: 25543205 Free PMC article.

6

Synthesis and evaluation of thymidine kinase 1-targeting carboranyl pyrimidine nucleoside analogs for boron neutron capture therapy of cancer.

Agarwal HK, Khalil A, Ishita K, Yang W, Nakkula RJ, Wu LC, Ali T, Tiwari R, Byun Y, Barth RF, Tjarks W. Agarwal HK, et al. Among authors: khalil a. Eur J Med Chem. 2015 Jul 15;100:197-209. doi: 10.1016/j.ejmech.2015.05.042. Epub 2015 May 27. Eur J Med Chem. 2015. PMID: 26087030 Free PMC article.

7

Synthesis and biological evaluation of aminothiazoles against Histoplasma capsulatum and Cryptococcus neoformans.

Ishita K, Stefanopoulos S, Khalil A, Cheng X, Tjarks W, Rappleye CA. Ishita K, et al. Among authors: khalil a. Bioorg Med Chem. 2018 May 15;26(9):2251-2261. doi: 10.1016/j.bmc.2018.01.024. Epub 2018 Feb 2. Bioorg Med Chem. 2018. PMID: 29580849 Free PMC article.

8

Discovery of new anticancer thiourea-azetidine hybrids: design, synthesis, in vitro antiproliferative, SAR, in silico molecular docking against VEGFR-2, ADMET, toxicity, and DFT studies.

Parmar DR, Soni JY, Guduru R, Rayani RH, Kusurkar RV, Vala AG, Talukdar SN, Eissa IH, Metwaly AM, Khalil A, Zunjar V, Battula S. Parmar DR, et al. Among authors: khalil a. Bioorg Chem. 2021 Oct;115:105206. doi: 10.1016/j.bioorg.2021.105206. Epub 2021 Jul 27. Bioorg Chem. 2021. PMID: 34339975

9

Nucleoside Scaffolds and Carborane Clusters for Boron Neutron Capture Therapy: Developments and Future Perspective.

Khalil A, Adam MSS. Khalil A, et al. Curr Med Chem. 2023 Oct 10. doi: 10.2174/0109298673245020230929152030. Online ahead of print. Curr Med Chem. 2023. PMID: 37818562

10

Rapid synthesis of 2',3'-dideoxy-3'β-fluoro-pyrimidine nucleosides from 2'-deoxypyrimidine nucleosides.

Khalil A, Mathé C, Périgaud C. Khalil A, et al. Bioorg Chem. 2010 Dec;38(6):271-4. doi: 10.1016/j.bioorg.2010.08.003. Epub 2010 Sep 7. Bioorg Chem. 2010. PMID: 20869741

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