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Structure-based design, parallel synthesis, structure-activity relationship, and molecular modeling studies of thiocarbamates, new potent non-nucleoside HIV-1 reverse transcriptase inhibitor isosteres of phenethylthiazolylthiourea derivatives.
Ranise A, Spallarossa A, Cesarini S, Bondavalli F, Schenone S, Bruno O, Menozzi G, Fossa P, Mosti L, La Colla M, Sanna G, Murreddu M, Collu G, Busonera B, Marongiu ME, Pani A, La Colla P, Loddo R. Ranise A, et al. J Med Chem. 2005 Jun 2;48(11):3858-73. doi: 10.1021/jm049252r. J Med Chem. 2005. PMID: 15916438
Assuming as a lead compound O-[2-(phthalimido)ethyl]phenylthiocarbamate 12, one of the precursors of the previously described acylthiocarbamates (Ranise, A.; et al. ...The lead optimization strategy led to para-substituted TCs 31, 33, 34, 39, 40, 41, 44, 45, …
Assuming as a lead compound O-[2-(phthalimido)ethyl]phenylthiocarbamate 12, one of the precursors of the previously described acylthi …
Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 1: Parallel synthesis, molecular modelling and structure-activity relationship studies on O-[2-(hetero)arylethyl]-N-phenylthiocarbamates.
Cesarini S, Spallarossa A, Ranise A, Fossa P, La Colla P, Sanna G, Collu G, Loddo R. Cesarini S, et al. Among authors: ranise a. Bioorg Med Chem. 2008 Apr 1;16(7):4160-72. doi: 10.1016/j.bmc.2007.12.050. Epub 2007 Dec 25. Bioorg Med Chem. 2008. PMID: 18226532
Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 2: Parallel synthesis, molecular modelling and structure-activity relationship studies on analogues of O-(2-phenylethyl)-N-phenylthiocarbamate.
Cesarini S, Spallarossa A, Ranise A, Bruno O, La Colla P, Secci B, Collu G, Loddo R. Cesarini S, et al. Among authors: ranise a. Bioorg Med Chem. 2008 Apr 1;16(7):4173-85. doi: 10.1016/j.bmc.2007.12.046. Epub 2007 Dec 25. Bioorg Med Chem. 2008. PMID: 18226533
Novel modifications in the series of O-(2-phthalimidoethyl)-N-substituted thiocarbamates and their ring-opened congeners as non-nucleoside HIV-1 reverse transcriptase inhibitors.
Spallarossa A, Cesarini S, Ranise A, Bruno O, Schenone S, La Colla P, Collu G, Sanna G, Secci B, Loddo R. Spallarossa A, et al. Among authors: ranise a. Eur J Med Chem. 2009 Apr;44(4):1650-63. doi: 10.1016/j.ejmech.2008.09.024. Epub 2008 Sep 30. Eur J Med Chem. 2009. PMID: 18954921
108 results