Tomassi C - Search Results

1

Progress in the design and development of phosphoinositide 3-kinase (PI3K) inhibitors for the treatment of chronic diseases.

Shuttleworth S, Silva F, Tomassi C, Cecil A, Hill T, Rogers H, Townsend P. Shuttleworth S, et al. Among authors: tomassi c. Prog Med Chem. 2009;48:81-131. doi: 10.1016/s0079-6468(09)04803-6. Prog Med Chem. 2009. PMID: 21544958 Review. No abstract available.

2

Progress in the preclinical discovery and clinical development of class I and dual class I/IV phosphoinositide 3-kinase (PI3K) inhibitors.

Shuttleworth SJ, Silva FA, Cecil AR, Tomassi CD, Hill TJ, Raynaud FI, Clarke PA, Workman P. Shuttleworth SJ, et al. Among authors: tomassi cd. Curr Med Chem. 2011;18(18):2686-714. doi: 10.2174/092986711796011229. Curr Med Chem. 2011. PMID: 21649578 Free PMC article. Review.

3

Progress in the development of small molecule therapeutics targeting Th17 cell function for the treatment of immune-inflammatory diseases.

Shuttleworth S, Townsend P, Silva F, Cecil A, Hill T, Tomassi C, Rogers H, Harrison R. Shuttleworth S, et al. Among authors: tomassi c. Prog Med Chem. 2011;50:109-33. doi: 10.1016/B978-0-12-381290-2.00003-3. Prog Med Chem. 2011. PMID: 21315929 No abstract available.

4

Disubstituted Bis-THF Moieties as New P2 Ligands in Nonpeptidal HIV-1 Protease Inhibitors.

Hohlfeld K, Tomassi C, Wegner JK, Kesteleyn B, Linclau B. Hohlfeld K, et al. Among authors: tomassi c. ACS Med Chem Lett. 2011 Mar 31;2(6):461-5. doi: 10.1021/ml2000356. eCollection 2011 Jun 9. ACS Med Chem Lett. 2011. PMID: 24900331 Free PMC article.

5

First synthesis and evaluation of the inhibitory effects of aza analogues of TSAO on HIV-1 replication.

Nguyen Van Nhien A, Tomassi C, Len C, Marco-Contelles JL, Balzarini J, Pannecouque C, De Clercq E, Postel D. Nguyen Van Nhien A, et al. Among authors: tomassi c. J Med Chem. 2005 Jun 30;48(13):4276-84. doi: 10.1021/jm050091g. J Med Chem. 2005. PMID: 15974581

6

Enantioselective synthesis and selective monofunctionalization of (4R,6R)-4,6- dihydroxy-2,8-dioxabicyclo[3.3.0]octane.

Linclau B, Jeffery MJ, Josse S, Tomassi C. Linclau B, et al. Among authors: tomassi c. Org Lett. 2006 Dec 7;8(25):5821-4. doi: 10.1021/ol062431d. Org Lett. 2006. PMID: 17134281

7

Synthesis and in vivo evaluation of 4-deoxy-4,4-difluoro-KRN7000.

Leung L, Tomassi C, Van Beneden K, Decruy T, Elewaut D, Elliott T, Al-Shamkhani A, Ottensmeier C, Van Calenbergh S, Werner J, Williams T, Linclau B. Leung L, et al. Among authors: tomassi c. Org Lett. 2008 Oct 16;10(20):4433-6. doi: 10.1021/ol801663m. Epub 2008 Sep 18. Org Lett. 2008. PMID: 18798635

8

The synthesis and in vivo evaluation of 2',2'-difluoro KRN7000.

Leung L, Tomassi C, Van Beneden K, Decruy T, Trappeniers M, Elewaut D, Gao Y, Elliott T, Al-Shamkhani A, Ottensmeier C, Werner JM, Williams A, Van Calenbergh S, Linclau B. Leung L, et al. Among authors: tomassi c. ChemMedChem. 2009 Mar;4(3):329-34. doi: 10.1002/cmdc.200800348. ChemMedChem. 2009. PMID: 19137519

9

Synthesis of AZA analogues of TSAO.

Nguyen Van Nhien A, Tomassi C, Len C, Marco-Contelles JL, Postel D. Nguyen Van Nhien A, et al. Among authors: tomassi c. Nucleosides Nucleotides Nucleic Acids. 2003 May-Aug;22(5-8):939-41. doi: 10.1081/NCN-120022690. Nucleosides Nucleotides Nucleic Acids. 2003. PMID: 14565316

10

Computational analysis of aza analogues of [2',5'-bis-O-(tert-butyldimethylsilyl)-beta-D-ribofuranose]-3'-spiro-5"-(4"-amino-1",2"-oxathiole-2",2"-dioxide) (TSAO) as HIV-1 reverse transcriptase inhibitors: relevance of conformational properties on the inhibitory activity.

Soriano E, Marco-Contelles J, Tomassi C, Nguyen Van Nhien A, Postel D. Soriano E, et al. Among authors: tomassi c. J Chem Inf Model. 2006 Jul-Aug;46(4):1666-77. doi: 10.1021/ci0600410. J Chem Inf Model. 2006. PMID: 16859298

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

15 results

Search Page