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Cardiac myosin activation: a potential therapeutic approach for systolic heart failure.
Science. 2011 Mar 18;331(6023):1439-43. doi: 10.1126/science.1200113.
Science. 2011.
PMID: 21415352
Free PMC article.
Activation of fast skeletal muscle troponin as a potential therapeutic approach for treating neuromuscular diseases.
Russell AJ, Hartman JJ, Hinken AC, Muci AR, Kawas R, Driscoll L, Godinez G, Lee KH, Marquez D, Browne WF 4th, Chen MM, Clarke D, Collibee SE, Garard M, Hansen R, Jia Z, Lu PP, Rodriguez H, Saikali KG, Schaletzky J, Vijayakumar V, Albertus DL, Claflin DR, Morgans DJ, Morgan BP, Malik FI.
Russell AJ, et al. Among authors: kawas r.
Nat Med. 2012 Feb 19;18(3):452-5. doi: 10.1038/nm.2618.
Nat Med. 2012.
PMID: 22344294
Free PMC article.
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A small-molecule modulator of cardiac myosin acts on multiple stages of the myosin chemomechanical cycle.
Kawas RF, Anderson RL, Ingle SRB, Song Y, Sran AS, Rodriguez HM.
Kawas RF, et al.
J Biol Chem. 2017 Oct 6;292(40):16571-16577. doi: 10.1074/jbc.M117.776815. Epub 2017 Aug 14.
J Biol Chem. 2017.
PMID: 28808052
Free PMC article.
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Discovery of omecamtiv mecarbil the first, selective, small molecule activator of cardiac Myosin.
Morgan BP, Muci A, Lu PP, Qian X, Tochimoto T, Smith WW, Garard M, Kraynack E, Collibee S, Suehiro I, Tomasi A, Valdez SC, Wang W, Jiang H, Hartman J, Rodriguez HM, Kawas R, Sylvester S, Elias KA, Godinez G, Lee K, Anderson R, Sueoka S, Xu D, Wang Z, Djordjevic N, Malik FI, Morgans DJ Jr.
Morgan BP, et al. Among authors: kawas r.
ACS Med Chem Lett. 2010 Aug 20;1(9):472-7. doi: 10.1021/ml100138q. eCollection 2010 Dec 9.
ACS Med Chem Lett. 2010.
PMID: 24900233
Free PMC article.
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A small-molecule inhibitor of sarcomere contractility suppresses hypertrophic cardiomyopathy in mice.
Green EM, Wakimoto H, Anderson RL, Evanchik MJ, Gorham JM, Harrison BC, Henze M, Kawas R, Oslob JD, Rodriguez HM, Song Y, Wan W, Leinwand LA, Spudich JA, McDowell RS, Seidman JG, Seidman CE.
Green EM, et al. Among authors: kawas r.
Science. 2016 Feb 5;351(6273):617-21. doi: 10.1126/science.aad3456.
Science. 2016.
PMID: 26912705
Free PMC article.
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Discovery of Tirasemtiv, the First Direct Fast Skeletal Muscle Troponin Activator.
Collibee SE, Bergnes G, Muci A, Browne WF 4th, Garard M, Hinken AC, Russell AJ, Suehiro I, Hartman J, Kawas R, Lu PP, Lee KH, Marquez D, Tomlinson M, Xu D, Kennedy A, Hwee D, Schaletzky J, Leung K, Malik FI, Morgans DJ Jr, Morgan BP.
Collibee SE, et al. Among authors: kawas r.
ACS Med Chem Lett. 2018 Feb 13;9(4):354-358. doi: 10.1021/acsmedchemlett.7b00546. eCollection 2018 Apr 12.
ACS Med Chem Lett. 2018.
PMID: 29670700
Free PMC article.
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