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Indazole derivatives as novel bradykinin B1 receptor antagonists.
Bioorg Med Chem Lett. 2010 Dec 1;20(23):7011-4. doi: 10.1016/j.bmcl.2010.09.121. Epub 2010 Sep 29.
Bioorg Med Chem Lett. 2010.
PMID: 20971001
Pyridine containing M(1) positive allosteric modulators with reduced plasma protein binding.
Kuduk SD, Di Marco CN, Cofre V, Pitts DR, Ray WJ, Ma L, Wittmann M, Seager MA, Koeplinger K, Thompson CD, Hartman GD, Bilodeau MT.
Kuduk SD, et al. Among authors: cofre v.
Bioorg Med Chem Lett. 2010 Jan 15;20(2):657-61. doi: 10.1016/j.bmcl.2009.11.059. Epub 2009 Dec 2.
Bioorg Med Chem Lett. 2010.
PMID: 19962304
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Fused heterocyclic M1 positive allosteric modulators.
Kuduk SD, Di Marco CN, Cofre V, Ray WJ, Ma L, Wittmann M, Seager MA, Koeplinger KA, Thompson CD, Hartman GD, Bilodeau MT.
Kuduk SD, et al. Among authors: cofre v.
Bioorg Med Chem Lett. 2011 May 1;21(9):2769-72. doi: 10.1016/j.bmcl.2010.10.028. Epub 2010 Oct 16.
Bioorg Med Chem Lett. 2011.
PMID: 21055928
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Amidine derived inhibitors of acid-sensing ion channel-3 (ASIC3).
Kuduk SD, Chang RK, Wai JM, Di Marco CN, Cofre V, DiPardo RM, Cook SP, Cato MJ, Jovanovska A, Urban MO, Leitl M, Spencer RH, Kane SA, Hartman GD, Bilodeau MT.
Kuduk SD, et al. Among authors: cofre v.
Bioorg Med Chem Lett. 2009 Aug 1;19(15):4059-63. doi: 10.1016/j.bmcl.2009.06.021. Epub 2009 Jun 13.
Bioorg Med Chem Lett. 2009.
PMID: 19553111
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N-heterocyclic derived M1 positive allosteric modulators.
Kuduk SD, Di Marco CN, Cofre V, Pitts DR, Ray WJ, Ma L, Wittmann M, Veng L, Seager MA, Koeplinger K, Thompson CD, Hartman GD, Bilodeau MT.
Kuduk SD, et al. Among authors: cofre v.
Bioorg Med Chem Lett. 2010 Feb 15;20(4):1334-7. doi: 10.1016/j.bmcl.2010.01.013. Epub 2010 Jan 11.
Bioorg Med Chem Lett. 2010.
PMID: 20097564
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α-Synuclein Drives Tau's Cytotoxic Aggregates Formation through Hydrophobic Interactions.
Ojeda A, Cofré V, Melo F, Caballero L, Fuentealba D, Cornejo A.
Ojeda A, et al. Among authors: cofre v.
Chempluschem. 2023 Oct;88(10):e202300257. doi: 10.1002/cplu.202300257. Epub 2023 Oct 4.
Chempluschem. 2023.
PMID: 37708459
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