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(1S)-1,5-anhydro-1-[5-(4-ethoxybenzyl)-2-methoxy-4-methylphenyl]-1-thio-D-glucitol (TS-071) is a potent, selective sodium-dependent glucose cotransporter 2 (SGLT2) inhibitor for type 2 diabetes treatment.
Kakinuma H, Oi T, Hashimoto-Tsuchiya Y, Arai M, Kawakita Y, Fukasawa Y, Iida I, Hagima N, Takeuchi H, Chino Y, Asami J, Okumura-Kitajima L, Io F, Yamamoto D, Miyata N, Takahashi T, Uchida S, Yamamoto K. Kakinuma H, et al. Among authors: fukasawa y. J Med Chem. 2010 Apr 22;53(8):3247-61. doi: 10.1021/jm901893x. J Med Chem. 2010. PMID: 20302302
In vitro and in vivo evaluation of the metabolism and bioavailability of ester prodrugs of mgs0039 (3-(3,4-dichlorobenzyloxy)-2-amino-6-fluorobicyclo[3.1.0]hexane-2,6-dicarboxylic Acid), a potent metabotropic glutamate receptor antagonist.
Nakamura M, Kawakita Y, Yasuhara A, Fukasawa Y, Yoshida K, Sakagami K, Nakazato A. Nakamura M, et al. Among authors: fukasawa y. Drug Metab Dispos. 2006 Mar;34(3):369-74. doi: 10.1124/dmd.105.006213. Epub 2005 Dec 2. Drug Metab Dispos. 2006. PMID: 16326817
Lymphopenia induced by a novel selective S1P(1) antagonist structurally unrelated to S1P.
Fujii Y, Ohtake H, Ono N, Hara T, Sakurai T, Takahashi S, Takayama T, Fukasawa Y, Shiozawa F, Tsukahara N, Hirayama T, Igarashi Y, Goitsuka R. Fujii Y, et al. Among authors: fukasawa y. Biochim Biophys Acta. 2012 Apr;1821(4):600-6. doi: 10.1016/j.bbalip.2011.12.006. Epub 2011 Dec 30. Biochim Biophys Acta. 2012. PMID: 22265714
186 results