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Exploration of SAR features by modifications of thiazoleacetic acids as CRTH2 antagonists.
Bioorg Med Chem Lett. 2010 Mar 1;20(5):1638-41. doi: 10.1016/j.bmcl.2010.01.092. Epub 2010 Jan 22.
Bioorg Med Chem Lett. 2010.
PMID: 20137942
Novel selective orally active CRTH2 antagonists for allergic inflammation developed from in silico derived hits.
Ulven T, Receveur JM, Grimstrup M, Rist Ø, Frimurer TM, Gerlach LO, Mathiesen JM, Kostenis E, Uller L, Högberg T.
Ulven T, et al. Among authors: grimstrup m.
J Med Chem. 2006 Nov 16;49(23):6638-41. doi: 10.1021/jm060657g.
J Med Chem. 2006.
PMID: 17154491
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Novel selective thiazoleacetic acids as CRTH2 antagonists developed from in silico derived hits. Part 2.
Grimstrup M, Rist Ø, Receveur JM, Frimurer TM, Ulven T, Mathiesen JM, Kostenis E, Högberg T.
Grimstrup M, et al.
Bioorg Med Chem Lett. 2010 Feb 1;20(3):1181-5. doi: 10.1016/j.bmcl.2009.12.015. Epub 2009 Dec 6.
Bioorg Med Chem Lett. 2010.
PMID: 20022749
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Novel selective thiazoleacetic acids as CRTH2 antagonists developed from in silico derived hits. Part 1.
Rist Ø, Grimstrup M, Receveur JM, Frimurer TM, Ulven T, Kostenis E, Högberg T.
Rist Ø, et al. Among authors: grimstrup m.
Bioorg Med Chem Lett. 2010 Feb 1;20(3):1177-80. doi: 10.1016/j.bmcl.2009.12.008. Epub 2009 Dec 4.
Bioorg Med Chem Lett. 2010.
PMID: 20031403
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Evaluation of spectral libraries and sample preparation for DIA-LC-MS analysis of host cell proteins: A case study of a bacterially expressed recombinant biopharmaceutical protein.
Heissel S, Bunkenborg J, Kristiansen MP, Holmbjerg AF, Grimstrup M, Mørtz E, Kofoed T, Højrup P.
Heissel S, et al. Among authors: grimstrup m.
Protein Expr Purif. 2018 Jul;147:69-77. doi: 10.1016/j.pep.2018.03.002. Epub 2018 Mar 9.
Protein Expr Purif. 2018.
PMID: 29526817
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