Martín-Fontecha M - Search Results

1

Benzimidazole derivatives as new serotonin 5-HT6 receptor antagonists. Molecular mechanisms of receptor inactivation.

de la Fuente T, Martín-Fontecha M, Sallander J, Benhamú B, Campillo M, Medina RA, Pellissier LP, Claeysen S, Dumuis A, Pardo L, López-Rodríguez ML. de la Fuente T, et al. J Med Chem. 2010 Feb 11;53(3):1357-69. doi: 10.1021/jm901672k. J Med Chem. 2010. PMID: 20078106

2

Development of endocannabinoid-based chemical probes for the study of cannabinoid receptors.

Martín-Couce L, Martín-Fontecha M, Capolicchio S, López-Rodríguez ML, Ortega-Gutiérrez S. Martín-Couce L, et al. J Med Chem. 2011 Jul 28;54(14):5265-9. doi: 10.1021/jm2004392. Epub 2011 Jun 27. J Med Chem. 2011. PMID: 21675776

3

New serotonin 5-HT(1A) receptor agonists with neuroprotective effect against ischemic cell damage.

Marco I, Valhondo M, Martín-Fontecha M, Vázquez-Villa H, Del Río J, Planas A, Sagredo O, Ramos JA, Torrecillas IR, Pardo L, Frechilla D, Benhamú B, López-Rodríguez ML. Marco I, et al. J Med Chem. 2011 Dec 8;54(23):7986-99. doi: 10.1021/jm2007886. Epub 2011 Nov 11. J Med Chem. 2011. PMID: 22029386

4

New serotonin 5-HT1A receptor agonists endowed with antinociceptive activity in vivo.

Valhondo M, Marco I, Martín-Fontecha M, Vázquez-Villa H, Ramos JA, Berkels R, Lauterbach T, Benhamú B, López-Rodríguez ML. Valhondo M, et al. J Med Chem. 2013 Oct 24;56(20):7851-61. doi: 10.1021/jm400766k. Epub 2013 Oct 8. J Med Chem. 2013. PMID: 24050112

5

Serotonin 5-HT6 receptor antagonists for the treatment of cognitive deficiency in Alzheimer's disease.

Benhamú B, Martín-Fontecha M, Vázquez-Villa H, Pardo L, López-Rodríguez ML. Benhamú B, et al. J Med Chem. 2014 Sep 11;57(17):7160-81. doi: 10.1021/jm5003952. Epub 2014 Jun 3. J Med Chem. 2014. PMID: 24850589 Review.

6

The extracellular entrance provides selectivity to serotonin 5-HT7 receptor antagonists with antidepressant-like behavior in vivo.

Medina RA, Vázquez-Villa H, Gómez-Tamayo JC, Benhamú B, Martín-Fontecha M, de la Fuente T, Caltabiano G, Hedlund PB, Pardo L, López-Rodríguez ML. Medina RA, et al. J Med Chem. 2014 Aug 14;57(15):6879-84. doi: 10.1021/jm500880c. Epub 2014 Aug 5. J Med Chem. 2014. PMID: 25073094

7

A new serotonin 5-HT₆ receptor antagonist with procognitive activity - Importance of a halogen bond interaction to stabilize the binding.

González-Vera JA, Medina RA, Martín-Fontecha M, Gonzalez A, de la Fuente T, Vázquez-Villa H, García-Cárceles J, Botta J, McCormick PJ, Benhamú B, Pardo L, López-Rodríguez ML. González-Vera JA, et al. Sci Rep. 2017 Jan 24;7:41293. doi: 10.1038/srep41293. Sci Rep. 2017. PMID: 28117458 Free PMC article.

8

Development of Fluorescent Ligands for the Human 5-HT1A Receptor.

Alonso D, Vázquez-Villa H, Gamo AM, Martínez-Esperón MF, Tortosa M, Viso A, Fernández de la Pradilla R, Junquera E, Aicart E, Martín-Fontecha M, Benhamú B, López-Rodríguez ML, Ortega-Gutiérrez S. Alonso D, et al. ACS Med Chem Lett. 2010 May 14;1(6):249-53. doi: 10.1021/ml100053y. eCollection 2010 Sep 9. ACS Med Chem Lett. 2010. PMID: 24900203 Free PMC article.

9

Chemoproteomic Approach to Explore the Target Profile of GPCR ligands: Application to 5-HT1A and 5-HT6 Receptors.

Gamo AM, González-Vera JA, Rueda-Zubiaurre A, Alonso D, Vázquez-Villa H, Martín-Couce L, Palomares Ó, López JA, Martín-Fontecha M, Benhamú B, López-Rodríguez ML, Ortega-Gutiérrez S. Gamo AM, et al. Chemistry. 2016 Jan 22;22(4):1313-21. doi: 10.1002/chem.201503101. Epub 2015 Nov 12. Chemistry. 2016. PMID: 26560738

10

A Potent Isoprenylcysteine Carboxylmethyltransferase (ICMT) Inhibitor Improves Survival in Ras-Driven Acute Myeloid Leukemia.

Marín-Ramos NI, Balabasquer M, Ortega-Nogales FJ, Torrecillas IR, Gil-Ordóñez A, Marcos-Ramiro B, Aguilar-Garrido P, Cushman I, Romero A, Medrano FJ, Gajate C, Mollinedo F, Philips MR, Campillo M, Gallardo M, Martín-Fontecha M, López-Rodríguez ML, Ortega-Gutiérrez S. Marín-Ramos NI, et al. Among authors: martin fontecha m. J Med Chem. 2019 Jul 11;62(13):6035-6046. doi: 10.1021/acs.jmedchem.9b00145. Epub 2019 Jun 19. J Med Chem. 2019. PMID: 31181882

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