Pasquini S - Search Results

1

The 4-quinolone-3-carboxylic acid motif as a multivalent scaffold in medicinal chemistry.

Mugnaini C, Pasquini S, Corelli F. Mugnaini C, et al. Among authors: pasquini s. Curr Med Chem. 2009;16(14):1746-67. doi: 10.2174/092986709788186156. Curr Med Chem. 2009. PMID: 19442143 Review.

2

The bioisosteric concept applied to cannabinoid ligands.

Mugnaini C, Pasquini S, Corelli F. Mugnaini C, et al. Among authors: pasquini s. Curr Med Chem. 2012;19(28):4794-815. doi: 10.2174/092986712803341575. Curr Med Chem. 2012. PMID: 22830341 Review.

3

Synthesis, cannabinoid receptor affinity, and molecular modeling studies of substituted 1-aryl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamides.

Silvestri R, Cascio MG, La Regina G, Piscitelli F, Lavecchia A, Brizzi A, Pasquini S, Botta M, Novellino E, Di Marzo V, Corelli F. Silvestri R, et al. Among authors: pasquini s. J Med Chem. 2008 Mar 27;51(6):1560-76. doi: 10.1021/jm070566z. Epub 2008 Feb 23. J Med Chem. 2008. PMID: 18293908

4

Investigations on the 4-quinolone-3-carboxylic acid motif. 1. Synthesis and structure-activity relationship of a class of human immunodeficiency virus type 1 integrase inhibitors.

Pasquini S, Mugnaini C, Tintori C, Botta M, Trejos A, Arvela RK, Larhed M, Witvrouw M, Michiels M, Christ F, Debyser Z, Corelli F. Pasquini S, et al. J Med Chem. 2008 Aug 28;51(16):5125-9. doi: 10.1021/jm8003784. Epub 2008 Jul 30. J Med Chem. 2008. PMID: 18665580

5

Investigations on the 4-quinolone-3-carboxylic acid motif. 2. Synthesis and structure-activity relationship of potent and selective cannabinoid-2 receptor agonists endowed with analgesic activity in vivo.

Pasquini S, Botta L, Semeraro T, Mugnaini C, Ligresti A, Palazzo E, Maione S, Di Marzo V, Corelli F. Pasquini S, et al. J Med Chem. 2008 Aug 28;51(16):5075-84. doi: 10.1021/jm800552f. Epub 2008 Aug 5. J Med Chem. 2008. PMID: 18680276

6

New resorcinol-anandamide "hybrids" as potent cannabinoid receptor ligands endowed with antinociceptive activity in vivo.

Brizzi A, Brizzi V, Cascio MG, Corelli F, Guida F, Ligresti A, Maione S, Martinelli A, Pasquini S, Tuccinardi T, Di Marzo V. Brizzi A, et al. Among authors: pasquini s. J Med Chem. 2009 Apr 23;52(8):2506-14. doi: 10.1021/jm8016255. J Med Chem. 2009. PMID: 19331413

7

Synthesis, cannabinoid receptor affinity, molecular modeling studies and in vivo pharmacological evaluation of new substituted 1-aryl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamides. 2. Effect of the 3-carboxamide substituent on the affinity and selectivity profile.

Silvestri R, Ligresti A, La Regina G, Piscitelli F, Gatti V, Brizzi A, Pasquini S, Lavecchia A, Allarà M, Fantini N, Carai MA, Novellino E, Colombo G, Di Marzo V, Corelli F. Silvestri R, et al. Among authors: pasquini s. Bioorg Med Chem. 2009 Aug 1;17(15):5549-64. doi: 10.1016/j.bmc.2009.06.027. Epub 2009 Jun 21. Bioorg Med Chem. 2009. PMID: 19595596

8

Rapid combinatorial access to a library of 1,5-disubstituted-3-indole-N-alkylacetamides as CB2 receptor ligands.

Pasquini S, Mugnaini C, Brizzi A, Ligresti A, Di Marzo V, Ghiron C, Corelli F. Pasquini S, et al. J Comb Chem. 2009 Sep-Oct;11(5):795-8. doi: 10.1021/cc9000955. J Comb Chem. 2009. PMID: 19694453 No abstract available.

9

Investigations on the 4-quinolone-3-carboxylic acid motif. 3. Synthesis, structure-affinity relationships, and pharmacological characterization of 6-substituted 4-quinolone-3-carboxamides as highly selective cannabinoid-2 receptor ligands.

Pasquini S, Ligresti A, Mugnaini C, Semeraro T, Cicione L, De Rosa M, Guida F, Luongo L, De Chiaro M, Cascio MG, Bolognini D, Marini P, Pertwee R, Maione S, Di Marzo V, Corelli F. Pasquini S, et al. J Med Chem. 2010 Aug 26;53(16):5915-28. doi: 10.1021/jm100123x. J Med Chem. 2010. PMID: 20718492

10

Three-dimensional quantitative structure-selectivity relationships analysis guided rational design of a highly selective ligand for the cannabinoid receptor 2.

Brogi S, Corelli F, Di Marzo V, Ligresti A, Mugnaini C, Pasquini S, Tafi A. Brogi S, et al. Among authors: pasquini s. Eur J Med Chem. 2011 Feb;46(2):547-55. doi: 10.1016/j.ejmech.2010.11.034. Epub 2010 Nov 27. Eur J Med Chem. 2011. PMID: 21183257

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

96 results

Search Page