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A quantitative analysis of kinase inhibitor selectivity.
Nat Biotechnol. 2008 Jan;26(1):127-32. doi: 10.1038/nbt1358.
Nat Biotechnol. 2008.
PMID: 18183025
4-Quinazolinyloxy-diaryl ureas as novel BRAFV600E inhibitors.
Holladay MW, Campbell BT, Rowbottom MW, Chao Q, Sprankle KG, Lai AG, Abraham S, Setti E, Faraoni R, Tran L, Armstrong RC, Gunawardane RN, Gardner MF, Cramer MD, Gitnick D, Ator MA, Dorsey BD, Ruggeri BR, Williams M, Bhagwat SS, James J.
Holladay MW, et al. Among authors: faraoni r.
Bioorg Med Chem Lett. 2011 Sep 15;21(18):5342-6. doi: 10.1016/j.bmcl.2011.07.019. Epub 2011 Jul 14.
Bioorg Med Chem Lett. 2011.
PMID: 21807507
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Identification of 1-(3-(6,7-dimethoxyquinazolin-4-yloxy)phenyl)-3-(5-(1,1,1-trifluoro-2-methylpropan-2-yl)isoxazol-3-yl)urea hydrochloride (CEP-32496), a highly potent and orally efficacious inhibitor of V-RAF murine sarcoma viral oncogene homologue B1 (BRAF) V600E.
Rowbottom MW, Faraoni R, Chao Q, Campbell BT, Lai AG, Setti E, Ezawa M, Sprankle KG, Abraham S, Tran L, Struss B, Gibney M, Armstrong RC, Gunawardane RN, Nepomuceno RR, Valenta I, Hua H, Gardner MF, Cramer MD, Gitnick D, Insko DE, Apuy JL, Jones-Bolin S, Ghose AK, Herbertz T, Ator MA, Dorsey BD, Ruggeri B, Williams M, Bhagwat S, James J, Holladay MW.
Rowbottom MW, et al. Among authors: faraoni r.
J Med Chem. 2012 Feb 9;55(3):1082-105. doi: 10.1021/jm2009925. Epub 2012 Jan 23.
J Med Chem. 2012.
PMID: 22168626
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CEP-32496: a novel orally active BRAF(V600E) inhibitor with selective cellular and in vivo antitumor activity.
James J, Ruggeri B, Armstrong RC, Rowbottom MW, Jones-Bolin S, Gunawardane RN, Dobrzanski P, Gardner MF, Zhao H, Cramer MD, Hunter K, Nepomuceno RR, Cheng M, Gitnick D, Yazdanian M, Insko DE, Ator MA, Apuy JL, Faraoni R, Dorsey BD, Williams M, Bhagwat SS, Holladay MW.
James J, et al. Among authors: faraoni r.
Mol Cancer Ther. 2012 Apr;11(4):930-41. doi: 10.1158/1535-7163.MCT-11-0645. Epub 2012 Feb 7.
Mol Cancer Ther. 2012.
PMID: 22319199
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Total synthesis and structural revision of vannusals A and B: synthesis of the originally assigned structure of vannusal B.
Nicolaou KC, Ortiz A, Zhang H, Dagneau P, Lanver A, Jennings MP, Arseniyadis S, Faraoni R, Lizos DE.
Nicolaou KC, et al. Among authors: faraoni r.
J Am Chem Soc. 2010 May 26;132(20):7138-52. doi: 10.1021/ja100740t.
J Am Chem Soc. 2010.
PMID: 20443561
Free PMC article.
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A catalytic asymmetric three-component 1,4-addition/aldol reaction: enantioselective synthesis of the spirocyclic system of vannusal A.
Nicolaou KC, Tang W, Dagneau P, Faraoni R.
Nicolaou KC, et al. Among authors: faraoni r.
Angew Chem Int Ed Engl. 2005 Jun 20;44(25):3874-9. doi: 10.1002/anie.200500789.
Angew Chem Int Ed Engl. 2005.
PMID: 15900527
No abstract available.
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New Rebek imide-type receptors for adenine featuring acetylene-linked pi-stacking platforms.
Faraoni R, Blanzat M, Kubicek S, Braun C, Schweizer WB, Gramlich V, Diederich F.
Faraoni R, et al.
Org Biomol Chem. 2004 Jul 21;2(14):1962-4. doi: 10.1039/b404311a. Epub 2004 Jun 10.
Org Biomol Chem. 2004.
PMID: 15254618
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H-Bonded complexes of adenine with Rebek imide receptors are stabilised by cation-pi interactions and destabilised by stacking with perfluoroaromatics.
Faraoni R, Castellano RK, Gramlich V, Diederich F.
Faraoni R, et al.
Chem Commun (Camb). 2004 Feb 21;(4):370-1. doi: 10.1039/b314353h. Epub 2004 Jan 23.
Chem Commun (Camb). 2004.
PMID: 14765213
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