Bilcer G - Search Results

1

Memapsin 2 (beta-secretase) inhibitor drug, between fantasy and reality.

Ghosh AK, Bilcer G, Hong L, Koelsch G, Tang J. Ghosh AK, et al. Among authors: bilcer g. Curr Alzheimer Res. 2007 Sep;4(4):418-22. doi: 10.2174/156720507781788864. Curr Alzheimer Res. 2007. PMID: 17908045 Review.

2

Structure-based design of cycloamide-urethane-derived novel inhibitors of human brain memapsin 2 (beta-secretase).

Ghosh AK, Devasamudram T, Hong L, DeZutter C, Xu X, Weerasena V, Koelsch G, Bilcer G, Tang J. Ghosh AK, et al. Among authors: bilcer g. Bioorg Med Chem Lett. 2005 Jan 3;15(1):15-20. doi: 10.1016/j.bmcl.2004.10.084. Bioorg Med Chem Lett. 2005. PMID: 15582402

3

Design, synthesis and X-ray structure of protein-ligand complexes: important insight into selectivity of memapsin 2 (beta-secretase) inhibitors.

Ghosh AK, Kumaragurubaran N, Hong L, Lei H, Hussain KA, Liu CF, Devasamudram T, Weerasena V, Turner R, Koelsch G, Bilcer G, Tang J. Ghosh AK, et al. Among authors: bilcer g. J Am Chem Soc. 2006 Apr 26;128(16):5310-1. doi: 10.1021/ja058636j. J Am Chem Soc. 2006. PMID: 16620080 Free PMC article.

4

Design, synthesis, and X-ray structure of potent memapsin 2 (beta-secretase) inhibitors with isophthalamide derivatives as the P2-P3-ligands.

Ghosh AK, Kumaragurubaran N, Hong L, Kulkarni SS, Xu X, Chang W, Weerasena V, Turner R, Koelsch G, Bilcer G, Tang J. Ghosh AK, et al. Among authors: bilcer g. J Med Chem. 2007 May 17;50(10):2399-407. doi: 10.1021/jm061338s. Epub 2007 Apr 14. J Med Chem. 2007. PMID: 17432843

5

Structure-based design: potent inhibitors of human brain memapsin 2 (beta-secretase).

Ghosh AK, Bilcer G, Harwood C, Kawahama R, Shin D, Hussain KA, Hong L, Loy JA, Nguyen C, Koelsch G, Ermolieff J, Tang J. Ghosh AK, et al. Among authors: bilcer g. J Med Chem. 2001 Aug 30;44(18):2865-8. doi: 10.1021/jm0101803. J Med Chem. 2001. PMID: 11520194

6

Structure-based design, synthesis and biological evaluation of novel β-secretase inhibitors containing a pyrazole or thiazole moiety as the P3 ligand.

Ghosh AK, Brindisi M, Yen YC, Xu X, Huang X, Devasamudram T, Bilcer G, Lei H, Koelsch G, Mesecar AD, Tang J. Ghosh AK, et al. Among authors: bilcer g. Bioorg Med Chem Lett. 2015 Feb 1;25(3):668-72. doi: 10.1016/j.bmcl.2014.11.087. Epub 2014 Dec 6. Bioorg Med Chem Lett. 2015. PMID: 25537272 Free PMC article.

7

In vivo inhibition of Abeta production by memapsin 2 (beta-secretase) inhibitors.

Chang WP, Koelsch G, Wong S, Downs D, Da H, Weerasena V, Gordon B, Devasamudram T, Bilcer G, Ghosh AK, Tang J. Chang WP, et al. Among authors: bilcer g. J Neurochem. 2004 Jun;89(6):1409-16. doi: 10.1111/j.1471-4159.2004.02452.x. J Neurochem. 2004. PMID: 15189343 Free article.

8

A stereoselective synthesis of (+)-boronolide.

Ghosh AK, Bilcer G. Ghosh AK, et al. Among authors: bilcer g. Tetrahedron Lett. 2000 Feb 12;41(7):1003-1006. doi: 10.1016/S0040-4039(99)02246-7. Epub 2000 Jun 22. Tetrahedron Lett. 2000. PMID: 30449906 Free PMC article.

9

Syntheses of FDA Approved HIV Protease Inhibitors.

Ghosh AK, Bilcer G, Schiltz G. Ghosh AK, et al. Among authors: bilcer g. Synthesis (Stuttg). 2001;2001(15):2203-2229. doi: 10.1055/s-2001-18434. Synthesis (Stuttg). 2001. PMID: 30393404 Free PMC article.

10

Tartaric Acid and Tartrates in the Synthesis of Bioactive Molecules.

Ghosh AK, Koltun ES, Bilcer G. Ghosh AK, et al. Among authors: bilcer g. Synthesis (Stuttg). 2001;2001(9):1281-1301. doi: 10.1055/s-2001-15217. Synthesis (Stuttg). 2001. PMID: 30393405 Free PMC article.

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