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Allosteric enhancers for A1 adenosine receptor.
Mini Rev Med Chem. 2007 Jun;7(6):559-69. doi: 10.2174/138955707780859459.
Mini Rev Med Chem. 2007.
PMID: 17584155
Review.
Microwave-assisted synthesis of thieno[2,3-c]pyridine derivatives as a new series of allosteric enhancers at the adenosine A(1) receptor.
Romagnoli R, Baraldi PG, Moorman AR, Iaconinoto MA, Carrion MD, Cara CL, Tabrizi MA, Preti D, Fruttarolo F, Baker SP, Varani K, Borea PA.
Romagnoli R, et al. Among authors: iaconinoto ma.
Bioorg Med Chem Lett. 2006 Nov 1;16(21):5530-3. doi: 10.1016/j.bmcl.2006.08.041. Epub 2006 Aug 22.
Bioorg Med Chem Lett. 2006.
PMID: 16931014
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Synthesis and biological evaluation of 2-amino-3-(4-chlorobenzoyl)-4-[N-(substituted) piperazin-1-yl]thiophenes as potent allosteric enhancers of the A1 adenosine receptor.
Romagnoli R, Baraldi PG, Carrion MD, Cara CL, Cruz-Lopez O, Iaconinoto MA, Preti D, Shryock JC, Moorman AR, Vincenzi F, Varani K, Andrea Borea P.
Romagnoli R, et al. Among authors: iaconinoto ma.
J Med Chem. 2008 Sep 25;51(18):5875-9. doi: 10.1021/jm800586p. Epub 2008 Aug 26.
J Med Chem. 2008.
PMID: 18729349
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Synthesis and preliminary biological evaluation of new anti-tubulin agents containing different benzoheterocycles.
Romagnoli R, Baraldi PG, Jung MK, Iaconinoto MA, Carrion MD, Remusat V, Preti D, Tabrizi MA, Francesca F, De Clercq E, Balzarini J, Hamel E.
Romagnoli R, et al. Among authors: iaconinoto ma.
Bioorg Med Chem Lett. 2005 Sep 15;15(18):4048-52. doi: 10.1016/j.bmcl.2005.06.022.
Bioorg Med Chem Lett. 2005.
PMID: 16005627
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Synthesis and biological activity of alpha-bromoacryloyl lexitropsin conjugates.
Romagnoli R, Baraldi PG, Iaconinoto MA, Carrion MD, Tabrizi MA, Gambari R, Borgatti M, Heilmann J.
Romagnoli R, et al. Among authors: iaconinoto ma.
Eur J Med Chem. 2005 Nov;40(11):1123-8. doi: 10.1016/j.ejmech.2005.05.003. Epub 2005 Jul 11.
Eur J Med Chem. 2005.
PMID: 16006014
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