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Page 1
Design and synthesis of hepatoselective, pyrrole-based HMG-CoA reductase inhibitors.
Bioorg Med Chem Lett. 2007 Aug 15;17(16):4538-44. doi: 10.1016/j.bmcl.2007.05.096. Epub 2007 Jun 6.
Bioorg Med Chem Lett. 2007.
PMID: 17574412
Synthesis and SAR of selective benzothiophene, benzofuran, and indole-based peroxisome proliferator-activated receptor delta agonists.
Filzen GF, Bratton L, Cheng XM, Erasga N, Geyer A, Lee C, Lu G, Pulaski J, Sorenson RJ, Unangst PC, Trivedi BK, Xu X.
Filzen GF, et al.
Bioorg Med Chem Lett. 2007 Jul 1;17(13):3630-5. doi: 10.1016/j.bmcl.2007.04.047. Epub 2007 Apr 24.
Bioorg Med Chem Lett. 2007.
PMID: 17512197
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Discovery of highly potent and selective benzyloxybenzyl-based peroxisome proliferator-activator receptor (PPAR) delta agonists.
Bratton LD, Filzen GF, Geyer A, Hoffman JK, Lu G, Pulaski J, Trivedi BK, Unangst PC, Xu X.
Bratton LD, et al.
Bioorg Med Chem Lett. 2007 Jul 1;17(13):3624-9. doi: 10.1016/j.bmcl.2007.04.046. Epub 2007 Apr 24.
Bioorg Med Chem Lett. 2007.
PMID: 17498950
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Discovery of pyrrole-based hepatoselective ligands as potent inhibitors of HMG-CoA reductase.
Bratton LD, Auerbach B, Choi C, Dillon L, Hanselman JC, Larsen SD, Lu G, Olsen K, Pfefferkorn JA, Robertson A, Sekerke C, Trivedi BK, Unangst PC.
Bratton LD, et al.
Bioorg Med Chem. 2007 Aug 15;15(16):5576-89. doi: 10.1016/j.bmc.2007.05.031. Epub 2007 May 17.
Bioorg Med Chem. 2007.
PMID: 17560788
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Thermodynamic and structure guided design of statin based inhibitors of 3-hydroxy-3-methylglutaryl coenzyme A reductase.
Sarver RW, Bills E, Bolton G, Bratton LD, Caspers NL, Dunbar JB, Harris MS, Hutchings RH, Kennedy RM, Larsen SD, Pavlovsky A, Pfefferkorn JA, Bainbridge G.
Sarver RW, et al. Among authors: bratton ld.
J Med Chem. 2008 Jul 10;51(13):3804-13. doi: 10.1021/jm7015057. Epub 2008 Jun 10.
J Med Chem. 2008.
PMID: 18540668
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Discovery of a series of 2-(1H-pyrazol-1-yl)pyridines as ALK5 inhibitors with potential utility in the prevention of dermal scarring.
Boys ML, Bian F, Kramer JB, Chio CL, Ren XD, Chen H, Barrett SD, Sexton KE, Iula DM, Filzen GF, Nguyen MN, Angell P, Downs VL, Wang Z, Raheja N, Ellsworth EL, Fakhoury S, Bratton LD, Keller PR, Gowan R, Drummond EM, Maiti SN, Hena MA, Lu L, McConnell P, Knafels JD, Thanabal V, Sun F, Alessi D, McCarthy A, Zhang E, Finzel BC, Patel S, Ciotti SM, Eisma R, Payne NA, Gilbertsen RB, Kostlan CR, Pocalyko DJ, Lala DS.
Boys ML, et al. Among authors: bratton ld.
Bioorg Med Chem Lett. 2012 May 15;22(10):3392-7. doi: 10.1016/j.bmcl.2012.04.013. Epub 2012 Apr 10.
Bioorg Med Chem Lett. 2012.
PMID: 22542194
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Quantitative measurement of JWH-018 and JWH-073 metabolites excreted in human urine.
Moran CL, Le VH, Chimalakonda KC, Smedley AL, Lackey FD, Owen SN, Kennedy PD, Endres GW, Ciske FL, Kramer JB, Kornilov AM, Bratton LD, Dobrowolski PJ, Wessinger WD, Fantegrossi WE, Prather PL, James LP, Radominska-Pandya A, Moran JH.
Moran CL, et al. Among authors: bratton ld.
Anal Chem. 2011 Jun 1;83(11):4228-36. doi: 10.1021/ac2005636. Epub 2011 May 6.
Anal Chem. 2011.
PMID: 21506519
Free PMC article.
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Biochemical characterization of alpha-ketooxadiazole inhibitors of elastases.
Wieczorek M, Gyorkos A, Spruce LW, Ettinger A, Ross SE, Kroona HS, Burgos-Lepley CE, Bratton LD, Drennan TS, Garnert DL, Von Burg G, Pilkington CG, Cheronis JC.
Wieczorek M, et al. Among authors: bratton ld.
Arch Biochem Biophys. 1999 Jul 15;367(2):193-201. doi: 10.1006/abbi.1999.1249.
Arch Biochem Biophys. 1999.
PMID: 10395735
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